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Compound Detail

CHEMBL1393195

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COc1cccc(-c2cc(O)c3cc(NC(=O)c4ccc(N(C)C)cc4)ccc3n2)c1

Basic Information

ChEMBL ID CHEMBL1393195
Phase Preclinical
Structure Type MOL
InChI Key NGOHFZIFIFSACZ-UHFFFAOYSA-N
2
Targets
8
Activities
2
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

413.5
MW (Da)
4.93
ALogP
5
HBA
2
HBD
74.7
PSA (Ų)
0.49
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C25H23N3O3
MW 413.48
Aromatic Rings 4
Heavy Atoms 31
NP-Likeness -1.23

Activity Summary

EC50 7 meas. best 6.53
IC50 1 meas. best 5.21

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
EC50 6.53 6.285 296.0 4
BJ
CHEMBL614358
EC50 6.18 6.1667 664.0 3
Unchecked
CHEMBL612545
IC50 5.21 5.21 6220.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine