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Compound Detail

CHEMBL1518905

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CCN1/C(=C\C=C\C2=[N+](CC)c3ccccc3C2(C)C)C(C)(C)c2ccccc21.[O-][Cl+3]([O-])([O-])[O-]

Basic Information

ChEMBL ID CHEMBL1518905
Phase Preclinical
Structure Type MOL
InChI Key MNCNXUGQOWTYOP-UHFFFAOYSA-M
Parent Compound CHEMBL1186511
Active Moiety CHEMBL1186511
9
Targets
15
Activities
2
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

385.6
MW (Da)
6.34
ALogP
1
HBA
0
HBD
6.2
PSA (Ų)
0.56
QED
1
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C27H33ClN2O4
MW 485.02
Aromatic Rings 2
Heavy Atoms 29
NP-Likeness -0.07

Activity Summary

EC50 11 meas. best 6.56
IC50 4 meas. best 7.19

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Sphingosine 1-phosphate receptor 2
CHEMBL2955
IC50 7.19 6.71 64.0 2
X-box-binding protein 1
CHEMBL1741176
IC50 6.8 6.8 160.0 1
BJ
CHEMBL614358
EC50 6.56 6.21 273.0 4
Unchecked
CHEMBL612545
EC50 6.04 6.04 903.0 1
Corticotropin-releasing factor receptor 2/Corticotropin-releasing factor-binding protein
CHEMBL3885546
EC50 5.43 5.43 3740.0 1
Streptococcus sp. 'group A'
CHEMBL612389
EC50 5.22 5.22 5963.0 1
Streptokinase A
CHEMBL1293228
EC50 5.13 4.97 7335.0 2
Streptococcus
CHEMBL612313
EC50 4.71 4.71 19539.0 1
Alkaline phosphatase, germ cell type
CHEMBL3402
IC50 4.66 4.66 22000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Sphingosine 1-phosphate receptor 2 IC50 = 64.0 nM 7.19 PUBCHEM_BIOASSAY: Counterscreen for S1P2 Antagonists: Dose Response Cell-Based S... -
X-box-binding protein 1 IC50 = 160.0 nM 6.8 PUBCHEM_BIOASSAY: XBP1 DR counterscreen for CHOP. (Class of assay: confirmatory)... -
BJ EC50 = 273.0 nM 6.56 PUBCHEM_BIOASSAY: Fluorescence Cell-Based Dose Response to Characterize Compound... -
BJ EC50 = 395.0 nM 6.4 PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Response HTS to Identify Compound... -
Sphingosine 1-phosphate receptor 2 IC50 = 587.0 nM 6.23 PUBCHEM_BIOASSAY: Dose Response Cell Based Assay for Antagonists of the S1P2 Rec... -
BJ EC50 = 664.0 nM 6.18 PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Confirmation HTS to Identify Comp... -
Unchecked EC50 = 903.0 nM 6.04 PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Response HTS to Identify Compound... -
BJ EC50 = 2006.0 nM 5.7 PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Response HTS to Identify Compound... -
Corticotropin-releasing factor receptor 2/Corticotropin-releasing factor-binding protein EC50 = 3740.0 nM 5.43 PUBCHEM_BIOASSAY: Dose Response confirmation of uHTS hits for small molecule ago... -
Streptococcus sp. 'group A' EC50 = 5963.0 nM 5.22 PUBCHEM_BIOASSAY: Luminescence Microorganism-Based Dose Confirmation HTS to Iden... -
Streptokinase A EC50 = 7335.0 nM 5.13 PUBCHEM_BIOASSAY: Luminescence Microorganism-Based Dose Confirmation HTS to Iden... -
Streptokinase A EC50 = 15637.0 nM 4.81 PUBCHEM_BIOASSAY: Absorbance Microorganism-Based Dose Response HTS to Identify I... -
Streptococcus EC50 = 19539.0 nM 4.71 PUBCHEM_BIOASSAY: Luminescence Microorganism-Based Dose Response HTS to Identify... -
Alkaline phosphatase, germ cell type IC50 = 22000.0 nM 4.66 PUBCHEM_BIOASSAY: Luminescent assay for HTS discovery of chemical inhibitors of ... -

Data from ChEMBL 36 via Core Engine