Assay Detail
Functional
CHEMBL1963988
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of uHTS hits for small molecule agonists of the CRF-binding protein and CRF-R2 receptor complex. (Class of assay: confirmatory)
2420
Total Activities
2420
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 6 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Target
Corticotropin-releasing factor receptor 2/Corticotropin-releasing factor-binding protein (CHEMBL3885546) ↗| Type | PROTEIN COMPLEX |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2420 | 5.12 | 6.34 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1995565 | — | — | 1 | 6.34 |
| CHEMBL1500274 | — | — | 1 | 6.26 |
| CHEMBL1464584 | — | — | 1 | 6.15 |
| CHEMBL1526609 | — | — | 1 | 6.10 |
| CHEMBL1519346 | — | — | 1 | 6.08 |
| CHEMBL1731330 | — | — | 1 | 6.06 |
| CHEMBL1720673 | — | — | 1 | 5.96 |
| CHEMBL1585011 | — | — | 1 | 5.95 |
| CHEMBL2001226 | — | — | 1 | 5.91 |
| CHEMBL1979183 | — | — | 1 | 5.86 |
| CHEMBL1530418 | — | — | 1 | 5.85 |
| CHEMBL1520994 | — | — | 1 | 5.78 |
| CHEMBL1707960 | — | — | 1 | 5.77 |
| CHEMBL1597458 | — | — | 1 | 5.74 |
| CHEMBL1334503 | — | — | 1 | 5.71 |
| CHEMBL1415013 | — | — | 1 | 5.71 |
| CHEMBL1730038 | — | — | 1 | 5.69 |
| CHEMBL1732456 | — | — | 1 | 5.68 |
| CHEMBL1347204 | — | — | 1 | 5.65 |
| CHEMBL1466606 | — | — | 1 | 5.64 |
| CHEMBL1590944 | — | — | 1 | 5.62 |
| CHEMBL1511951 | — | — | 1 | 5.61 |
| CHEMBL1502602 | — | — | 1 | 5.61 |
| CHEMBL1565644 | — | — | 1 | 5.59 |
| CHEMBL1888697 | — | — | 1 | 5.59 |
| CHEMBL1598335 | — | — | 1 | 5.59 |
| CHEMBL1370848 | — | — | 1 | 5.58 |
| CHEMBL1556958 | STROBOPININ | — | 1 | 5.57 |
| CHEMBL1873465 | — | — | 1 | 5.56 |
| CHEMBL1563791 | — | — | 1 | 5.56 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1995565 | — | EC50 | = | 460.0 | nM | 6.34 |
| CHEMBL1500274 | — | EC50 | = | 544.0 | nM | 6.26 |
| CHEMBL1464584 | — | EC50 | = | 709.0 | nM | 6.15 |
| CHEMBL1526609 | — | EC50 | = | 793.0 | nM | 6.10 |
| CHEMBL1519346 | — | EC50 | = | 832.0 | nM | 6.08 |
| CHEMBL1731330 | — | EC50 | = | 870.0 | nM | 6.06 |
| CHEMBL1720673 | — | EC50 | = | 1110.0 | nM | 5.96 |
| CHEMBL1585011 | — | EC50 | = | 1120.0 | nM | 5.95 |
| CHEMBL2001226 | — | EC50 | = | 1240.0 | nM | 5.91 |
| CHEMBL1979183 | — | EC50 | = | 1370.0 | nM | 5.86 |
| CHEMBL1530418 | — | EC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL1520994 | — | EC50 | = | 1650.0 | nM | 5.78 |
| CHEMBL1707960 | — | EC50 | = | 1690.0 | nM | 5.77 |
| CHEMBL1597458 | — | EC50 | = | 1830.0 | nM | 5.74 |
| CHEMBL1415013 | — | EC50 | = | 1970.0 | nM | 5.71 |
| CHEMBL1334503 | — | EC50 | = | 1970.0 | nM | 5.71 |
| CHEMBL1730038 | — | EC50 | = | 2050.0 | nM | 5.69 |
| CHEMBL1732456 | — | EC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL1347204 | — | EC50 | = | 2260.0 | nM | 5.65 |
| CHEMBL1466606 | — | EC50 | = | 2290.0 | nM | 5.64 |
| CHEMBL1590944 | — | EC50 | = | 2380.0 | nM | 5.62 |
| CHEMBL1511951 | — | EC50 | = | 2450.0 | nM | 5.61 |
| CHEMBL1502602 | — | EC50 | = | 2430.0 | nM | 5.61 |
| CHEMBL1888697 | — | EC50 | = | 2560.0 | nM | 5.59 |
| CHEMBL1565644 | — | EC50 | = | 2560.0 | nM | 5.59 |
| CHEMBL1598335 | — | EC50 | = | 2540.0 | nM | 5.59 |
| CHEMBL1370848 | — | EC50 | = | 2650.0 | nM | 5.58 |
| CHEMBL1556958 | STROBOPININ | EC50 | = | 2690.0 | nM | 5.57 |
| CHEMBL1563791 | — | EC50 | = | 2780.0 | nM | 5.56 |
| CHEMBL1589419 | — | EC50 | = | 2770.0 | nM | 5.56 |
| CHEMBL1310585 | — | EC50 | = | 2740.0 | nM | 5.56 |
| CHEMBL1873465 | — | EC50 | = | 2730.0 | nM | 5.56 |
| CHEMBL1409207 | — | EC50 | = | 2760.0 | nM | 5.56 |
| CHEMBL1977384 | — | EC50 | = | 2800.0 | nM | 5.55 |
| CHEMBL1715537 | — | EC50 | = | 2840.0 | nM | 5.55 |
| CHEMBL1415999 | — | EC50 | = | 2870.0 | nM | 5.54 |
| CHEMBL1421625 | — | EC50 | = | 2890.0 | nM | 5.54 |
| CHEMBL1524179 | — | EC50 | = | 2960.0 | nM | 5.53 |
| CHEMBL1419598 | — | EC50 | = | 3060.0 | nM | 5.51 |
| CHEMBL1510679 | — | EC50 | = | 3140.0 | nM | 5.50 |
| CHEMBL1894760 | — | EC50 | = | 3200.0 | nM | 5.50 |
| CHEMBL1429578 | — | EC50 | = | 3220.0 | nM | 5.49 |
| CHEMBL1424360 | — | EC50 | = | 3320.0 | nM | 5.48 |
| CHEMBL1527735 | — | EC50 | = | 3530.0 | nM | 5.45 |
| CHEMBL1518905 | — | EC50 | = | 3740.0 | nM | 5.43 |
| CHEMBL1733538 | — | EC50 | = | 3840.0 | nM | 5.42 |
| CHEMBL1484830 | — | EC50 | = | 3770.0 | nM | 5.42 |
| CHEMBL2005694 | — | EC50 | = | 3840.0 | nM | 5.42 |
| CHEMBL1720455 | — | EC50 | = | 3940.0 | nM | 5.41 |
| CHEMBL1495386 | — | EC50 | = | 3910.0 | nM | 5.41 |