Assay Detail
Functional
CHEMBL1614165
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Image-Based HTS for Selective Antagonists for GPR55. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2026, AID2809, AID2814, AID2815, AID2820, AID2822, AID2835, AID2836, AID485277, AID485278, AID485282, AID485283, AID485285, AID485286, AID485287, AID488947]
277
Total Activities
277
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 277 | 5.59 | 6.29 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1492859 | — | — | 1 | 6.29 |
| CHEMBL1349766 | — | — | 1 | 6.26 |
| CHEMBL1421591 | — | — | 1 | 6.26 |
| CHEMBL3198389 | — | — | 1 | 6.25 |
| CHEMBL1611658 | — | — | 1 | 6.23 |
| CHEMBL1495714 | — | — | 1 | 6.23 |
| CHEMBL1518491 | — | — | 1 | 6.22 |
| CHEMBL1367120 | — | — | 1 | 6.20 |
| CHEMBL1360615 | — | — | 1 | 6.18 |
| CHEMBL1313003 | — | — | 1 | 6.18 |
| CHEMBL1484306 | — | — | 1 | 6.18 |
| CHEMBL1410009 | — | — | 1 | 6.17 |
| CHEMBL1400386 | — | — | 1 | 6.17 |
| CHEMBL1542168 | — | — | 1 | 6.17 |
| CHEMBL1425137 | — | — | 1 | 6.16 |
| CHEMBL1366942 | — | — | 1 | 6.16 |
| CHEMBL1401308 | — | — | 1 | 6.11 |
| CHEMBL1353797 | — | — | 1 | 6.10 |
| CHEMBL1309286 | — | — | 1 | 6.10 |
| CHEMBL1413436 | — | — | 1 | 6.08 |
| CHEMBL1341584 | — | — | 1 | 6.08 |
| CHEMBL1324005 | — | — | 1 | 6.07 |
| CHEMBL1448070 | — | — | 1 | 6.06 |
| CHEMBL1469184 | — | — | 1 | 6.05 |
| CHEMBL942 | BISACODYL | 4.0 | 1 | 6.04 |
| CHEMBL1431310 | — | — | 1 | 6.04 |
| CHEMBL1431953 | — | — | 1 | 6.04 |
| CHEMBL1379600 | — | — | 1 | 6.02 |
| CHEMBL1452186 | — | — | 1 | 6.01 |
| CHEMBL1323770 | — | — | 1 | 6.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1492859 | — | IC50 | = | 508.61 | nM | 6.29 |
| CHEMBL1421591 | — | IC50 | = | 552.48 | nM | 6.26 |
| CHEMBL1349766 | — | IC50 | = | 542.66 | nM | 6.26 |
| CHEMBL3198389 | — | IC50 | = | 558.48 | nM | 6.25 |
| CHEMBL1495714 | — | IC50 | = | 587.26 | nM | 6.23 |
| CHEMBL1611658 | — | IC50 | = | 591.63 | nM | 6.23 |
| CHEMBL1518491 | — | IC50 | = | 598.02 | nM | 6.22 |
| CHEMBL1367120 | — | IC50 | = | 624.47 | nM | 6.20 |
| CHEMBL1360615 | — | IC50 | = | 664.95 | nM | 6.18 |
| CHEMBL1313003 | — | IC50 | = | 653.29 | nM | 6.18 |
| CHEMBL1484306 | — | IC50 | = | 653.47 | nM | 6.18 |
| CHEMBL1400386 | — | IC50 | = | 672.41 | nM | 6.17 |
| CHEMBL1410009 | — | IC50 | = | 678.23 | nM | 6.17 |
| CHEMBL1542168 | — | IC50 | = | 679.78 | nM | 6.17 |
| CHEMBL1366942 | — | IC50 | = | 699.18 | nM | 6.16 |
| CHEMBL1425137 | — | IC50 | = | 696.1 | nM | 6.16 |
| CHEMBL1401308 | — | IC50 | = | 768.58 | nM | 6.11 |
| CHEMBL1309286 | — | IC50 | = | 793.27 | nM | 6.10 |
| CHEMBL1353797 | — | IC50 | = | 798.71 | nM | 6.10 |
| CHEMBL1413436 | — | IC50 | = | 824.96 | nM | 6.08 |
| CHEMBL1341584 | — | IC50 | = | 824.1 | nM | 6.08 |
| CHEMBL1324005 | — | IC50 | = | 847.3 | nM | 6.07 |
| CHEMBL1448070 | — | IC50 | = | 868.6 | nM | 6.06 |
| CHEMBL1469184 | — | IC50 | = | 893.61 | nM | 6.05 |
| CHEMBL942 | BISACODYL | IC50 | = | 908.43 | nM | 6.04 |
| CHEMBL1431953 | — | IC50 | = | 914.99 | nM | 6.04 |
| CHEMBL1431310 | — | IC50 | = | 908.02 | nM | 6.04 |
| CHEMBL1379600 | — | IC50 | = | 964.6 | nM | 6.02 |
| CHEMBL1323770 | — | IC50 | = | 968.53 | nM | 6.01 |
| CHEMBL1452186 | — | IC50 | = | 978.34 | nM | 6.01 |
| CHEMBL1334080 | — | IC50 | = | 1081.87 | nM | 5.97 |
| CHEMBL1449992 | — | IC50 | = | 1059.65 | nM | 5.97 |
| CHEMBL1383283 | — | IC50 | = | 1070.62 | nM | 5.97 |
| CHEMBL1427618 | — | IC50 | = | 1083.31 | nM | 5.96 |
| CHEMBL1575373 | — | IC50 | = | 1084.61 | nM | 5.96 |
| CHEMBL1329450 | — | IC50 | = | 1124.93 | nM | 5.95 |
| CHEMBL1585390 | — | IC50 | = | 1113.43 | nM | 5.95 |
| CHEMBL1543720 | — | IC50 | = | 1115.35 | nM | 5.95 |
| CHEMBL1341792 | — | IC50 | = | 1178.44 | nM | 5.93 |
| CHEMBL1346587 | — | IC50 | = | 1177.99 | nM | 5.93 |
| CHEMBL1566398 | — | IC50 | = | 1165.59 | nM | 5.93 |
| CHEMBL1480330 | — | IC50 | = | 1203.1 | nM | 5.92 |
| CHEMBL1499761 | — | IC50 | = | 1202.85 | nM | 5.92 |
| CHEMBL1411212 | — | IC50 | = | 1235.98 | nM | 5.91 |
| CHEMBL1457590 | — | IC50 | = | 1219.18 | nM | 5.91 |
| CHEMBL1491374 | — | IC50 | = | 1249.07 | nM | 5.90 |
| CHEMBL1452926 | — | IC50 | = | 1267.66 | nM | 5.90 |
| CHEMBL1466203 | — | IC50 | = | 1259.18 | nM | 5.90 |
| CHEMBL1466352 | — | IC50 | = | 1312.01 | nM | 5.88 |
| CHEMBL417727 | — | IC50 | = | 1364.05 | nM | 5.87 |