Assay Detail
Functional
CHEMBL1614201
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Confirmation HTS to Identify Inhibitors of Platelet Dense Granule Release. (Class of assay: confirmatory) [Related pubchem assays: 1663 (Primary HTS), 1678 (Summary of Project)]
1584
Total Activities
1584
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1584 | 5.29 | 6.94 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1443750 | — | — | 1 | 6.94 |
| CHEMBL1417508 | — | — | 1 | 6.90 |
| CHEMBL1975118 | — | — | 1 | 6.87 |
| CHEMBL1980658 | — | — | 1 | 6.86 |
| CHEMBL1612044 | — | — | 1 | 6.84 |
| CHEMBL1386646 | — | — | 1 | 6.83 |
| CHEMBL1973921 | — | — | 1 | 6.81 |
| CHEMBL3199673 | — | — | 1 | 6.77 |
| CHEMBL1994596 | — | — | 1 | 6.76 |
| CHEMBL405317 | — | — | 1 | 6.72 |
| CHEMBL1459468 | — | — | 1 | 6.71 |
| CHEMBL1509670 | — | — | 1 | 6.69 |
| CHEMBL1383312 | — | — | 1 | 6.68 |
| CHEMBL3196469 | — | — | 1 | 6.68 |
| CHEMBL1256672 | — | — | 1 | 6.65 |
| CHEMBL260342 | — | — | 1 | 6.64 |
| CHEMBL1539359 | — | — | 1 | 6.63 |
| CHEMBL339304 | — | — | 1 | 6.63 |
| CHEMBL1301576 | — | — | 1 | 6.62 |
| CHEMBL1511219 | — | — | 1 | 6.62 |
| CHEMBL1557637 | — | — | 1 | 6.60 |
| CHEMBL1928491 | — | — | 1 | 6.59 |
| CHEMBL1965132 | — | — | 1 | 6.53 |
| CHEMBL2007273 | — | — | 1 | 6.50 |
| CHEMBL1467431 | — | — | 1 | 6.48 |
| CHEMBL1484327 | — | — | 1 | 6.47 |
| CHEMBL1524484 | — | — | 1 | 6.45 |
| CHEMBL1595632 | — | — | 1 | 6.44 |
| CHEMBL1581417 | — | — | 1 | 6.44 |
| CHEMBL3192393 | — | — | 1 | 6.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1443750 | — | EC50 | = | 115.0 | nM | 6.94 |
| CHEMBL1417508 | — | EC50 | = | 125.0 | nM | 6.90 |
| CHEMBL1975118 | — | EC50 | = | 136.0 | nM | 6.87 |
| CHEMBL1980658 | — | EC50 | = | 138.0 | nM | 6.86 |
| CHEMBL1612044 | — | EC50 | = | 144.0 | nM | 6.84 |
| CHEMBL1386646 | — | EC50 | = | 149.0 | nM | 6.83 |
| CHEMBL1973921 | — | EC50 | = | 156.0 | nM | 6.81 |
| CHEMBL3199673 | — | EC50 | = | 170.0 | nM | 6.77 |
| CHEMBL1994596 | — | EC50 | = | 172.0 | nM | 6.76 |
| CHEMBL405317 | — | EC50 | = | 189.0 | nM | 6.72 |
| CHEMBL1459468 | — | EC50 | = | 196.0 | nM | 6.71 |
| CHEMBL1509670 | — | EC50 | = | 205.0 | nM | 6.69 |
| CHEMBL1383312 | — | EC50 | = | 208.0 | nM | 6.68 |
| CHEMBL3196469 | — | EC50 | = | 209.0 | nM | 6.68 |
| CHEMBL1256672 | — | EC50 | = | 224.0 | nM | 6.65 |
| CHEMBL260342 | — | EC50 | = | 231.0 | nM | 6.64 |
| CHEMBL339304 | — | EC50 | = | 235.0 | nM | 6.63 |
| CHEMBL1539359 | — | EC50 | = | 234.0 | nM | 6.63 |
| CHEMBL1301576 | — | EC50 | = | 240.0 | nM | 6.62 |
| CHEMBL1511219 | — | EC50 | = | 240.0 | nM | 6.62 |
| CHEMBL1557637 | — | EC50 | = | 250.0 | nM | 6.60 |
| CHEMBL1928491 | — | EC50 | = | 254.0 | nM | 6.59 |
| CHEMBL1965132 | — | EC50 | = | 298.0 | nM | 6.53 |
| CHEMBL2007273 | — | EC50 | = | 317.0 | nM | 6.50 |
| CHEMBL1467431 | — | EC50 | = | 333.0 | nM | 6.48 |
| CHEMBL1484327 | — | EC50 | = | 335.0 | nM | 6.47 |
| CHEMBL1524484 | — | EC50 | = | 352.0 | nM | 6.45 |
| CHEMBL1595632 | — | EC50 | = | 365.0 | nM | 6.44 |
| CHEMBL1581417 | — | EC50 | = | 361.0 | nM | 6.44 |
| CHEMBL3192393 | — | EC50 | = | 407.0 | nM | 6.39 |
| CHEMBL1392570 | — | EC50 | = | 429.0 | nM | 6.37 |
| CHEMBL1327810 | — | EC50 | = | 435.0 | nM | 6.36 |
| CHEMBL1519965 | — | EC50 | = | 443.0 | nM | 6.35 |
| CHEMBL1533835 | — | EC50 | = | 457.0 | nM | 6.34 |
| CHEMBL408850 | — | EC50 | = | 468.0 | nM | 6.33 |
| CHEMBL1330058 | — | EC50 | = | 475.0 | nM | 6.32 |
| CHEMBL1450797 | — | EC50 | = | 499.0 | nM | 6.30 |
| CHEMBL1495092 | — | EC50 | = | 504.0 | nM | 6.30 |
| CHEMBL3194013 | — | EC50 | = | 533.0 | nM | 6.27 |
| CHEMBL3211930 | — | EC50 | = | 564.0 | nM | 6.25 |
| CHEMBL1335571 | — | EC50 | = | 623.0 | nM | 6.21 |
| CHEMBL1462373 | — | EC50 | = | 621.0 | nM | 6.21 |
| CHEMBL189 | MILRINONE | EC50 | = | 634.0 | nM | 6.20 |
| CHEMBL3197960 | — | EC50 | = | 693.0 | nM | 6.16 |
| CHEMBL1361038 | — | EC50 | = | 706.0 | nM | 6.15 |
| CHEMBL1200759 | ANAGRELIDE HYDROCHLORIDE | EC50 | = | 722.0 | nM | 6.14 |
| CHEMBL530609 | — | EC50 | = | 738.0 | nM | 6.13 |
| CHEMBL1492671 | — | EC50 | = | 749.0 | nM | 6.13 |
| CHEMBL1306132 | — | EC50 | = | 738.0 | nM | 6.13 |
| CHEMBL477 | ADENOSINE | EC50 | = | 759.0 | nM | 6.12 |