Assay Detail
Functional
CHEMBL1614266
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: A High Throughput Confirmatory Assay used to Identify Novel Compounds that Inhibit Mycobacterium Tuberculosis in the absence of Glycerol. (Class of assay: confirmatory)
1732
Total Activities
1732
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1732 | 4.80 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1605956 | — | — | 1 | 6.70 |
| CHEMBL518923 | — | — | 1 | 6.70 |
| CHEMBL1344225 | — | — | 1 | 6.70 |
| CHEMBL3197433 | — | — | 1 | 6.70 |
| CHEMBL1345018 | — | — | 1 | 6.70 |
| CHEMBL1427913 | — | — | 1 | 6.70 |
| CHEMBL1410618 | — | — | 1 | 6.70 |
| CHEMBL3214555 | — | — | 1 | 6.70 |
| CHEMBL1368213 | — | — | 1 | 6.70 |
| CHEMBL1526067 | — | — | 1 | 6.70 |
| CHEMBL1550076 | — | — | 1 | 6.70 |
| CHEMBL1605089 | — | — | 1 | 6.70 |
| CHEMBL1512296 | — | — | 1 | 6.62 |
| CHEMBL1417731 | — | — | 1 | 6.38 |
| CHEMBL1378668 | — | — | 1 | 6.35 |
| CHEMBL1592492 | — | — | 1 | 6.35 |
| CHEMBL1966872 | — | — | 1 | 6.34 |
| CHEMBL1369671 | — | — | 1 | 6.30 |
| CHEMBL508338 | THIMEROSAL | 3.0 | 1 | 6.28 |
| CHEMBL1558514 | — | — | 1 | 6.22 |
| CHEMBL1405262 | — | — | 1 | 6.17 |
| CHEMBL1339324 | — | — | 1 | 6.14 |
| CHEMBL1543899 | — | — | 1 | 6.14 |
| CHEMBL478120 | MARBOFLOXACIN | 2.0 | 1 | 6.14 |
| CHEMBL1373411 | — | — | 1 | 6.13 |
| CHEMBL3196253 | — | — | 1 | 6.12 |
| CHEMBL1576407 | — | — | 1 | 6.09 |
| CHEMBL1389533 | — | — | 1 | 6.09 |
| CHEMBL1557632 | — | — | 1 | 6.02 |
| CHEMBL530038 | — | — | 1 | 6.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1605089 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1550076 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1427913 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1344225 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL3197433 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1605956 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1368213 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL518923 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL3214555 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1526067 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1410618 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1345018 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1512296 | — | IC50 | = | 240.0 | nM | 6.62 |
| CHEMBL1417731 | — | IC50 | = | 420.0 | nM | 6.38 |
| CHEMBL1592492 | — | IC50 | = | 450.0 | nM | 6.35 |
| CHEMBL1378668 | — | IC50 | = | 450.0 | nM | 6.35 |
| CHEMBL1966872 | — | IC50 | = | 460.0 | nM | 6.34 |
| CHEMBL1369671 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL508338 | THIMEROSAL | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL1558514 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL1405262 | — | IC50 | = | 670.0 | nM | 6.17 |
| CHEMBL1339324 | — | IC50 | = | 730.0 | nM | 6.14 |
| CHEMBL478120 | MARBOFLOXACIN | IC50 | = | 720.0 | nM | 6.14 |
| CHEMBL1543899 | — | IC50 | = | 730.0 | nM | 6.14 |
| CHEMBL1373411 | — | IC50 | = | 740.0 | nM | 6.13 |
| CHEMBL3196253 | — | IC50 | = | 750.0 | nM | 6.12 |
| CHEMBL1576407 | — | IC50 | = | 810.0 | nM | 6.09 |
| CHEMBL1389533 | — | IC50 | = | 820.0 | nM | 6.09 |
| CHEMBL1557632 | — | IC50 | = | 950.0 | nM | 6.02 |
| CHEMBL530038 | — | IC50 | = | 970.0 | nM | 6.01 |
| CHEMBL1359688 | — | IC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL1353054 | — | IC50 | = | 1090.0 | nM | 5.96 |
| CHEMBL461579 | — | IC50 | = | 1130.0 | nM | 5.95 |
| CHEMBL1497838 | — | IC50 | = | 1160.0 | nM | 5.94 |
| CHEMBL1995800 | — | IC50 | = | 1190.0 | nM | 5.92 |
| CHEMBL1502870 | — | IC50 | = | 1260.0 | nM | 5.90 |
| CHEMBL1606685 | — | IC50 | = | 1280.0 | nM | 5.89 |
| CHEMBL3199620 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL1448732 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL1427476 | — | IC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL1502273 | — | IC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL19954 | — | IC50 | = | 1330.0 | nM | 5.88 |
| CHEMBL1556750 | — | IC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL1543127 | — | IC50 | = | 1360.0 | nM | 5.87 |
| CHEMBL1472263 | — | IC50 | = | 1380.0 | nM | 5.86 |
| CHEMBL1341756 | — | IC50 | = | 1420.0 | nM | 5.85 |
| CHEMBL375781 | NEOCUPROINE | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL964 | DISULFIRAM | IC50 | = | 1460.0 | nM | 5.84 |
| CHEMBL1556481 | — | IC50 | = | 1430.0 | nM | 5.84 |
| CHEMBL1525222 | — | IC50 | = | 1490.0 | nM | 5.83 |