Assay Detail
Functional
CHEMBL1614289
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: High Throughput Screening Assay used to Identify Novel Compounds that Inhibit Mycobacterium Tuberculosis in 7H9 Media. (Class of assay: confirmatory)
1938
Total Activities
1938
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1938 | 4.87 | 6.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1313588 | — | — | 1 | 6.68 |
| CHEMBL1543899 | — | — | 1 | 6.58 |
| CHEMBL1494293 | — | — | 1 | 6.55 |
| CHEMBL1339324 | — | — | 1 | 6.52 |
| CHEMBL1340776 | — | — | 1 | 6.48 |
| CHEMBL508338 | THIMEROSAL | 3.0 | 1 | 6.47 |
| CHEMBL1562086 | — | — | 1 | 6.47 |
| CHEMBL1467760 | — | — | 1 | 6.47 |
| CHEMBL1417731 | — | — | 1 | 6.44 |
| CHEMBL1335703 | — | — | 1 | 6.43 |
| CHEMBL1407492 | — | — | 1 | 6.43 |
| CHEMBL1542899 | — | — | 1 | 6.42 |
| CHEMBL1373411 | — | — | 1 | 6.42 |
| CHEMBL1341756 | — | — | 1 | 6.41 |
| CHEMBL1303785 | — | — | 1 | 6.37 |
| CHEMBL1543127 | — | — | 1 | 6.32 |
| CHEMBL375781 | NEOCUPROINE | — | 1 | 6.31 |
| CHEMBL1396156 | — | — | 1 | 6.31 |
| CHEMBL1453396 | — | — | 1 | 6.29 |
| CHEMBL1556750 | — | — | 1 | 6.28 |
| CHEMBL1502870 | — | — | 1 | 6.28 |
| CHEMBL1420009 | — | — | 1 | 6.27 |
| CHEMBL1980982 | — | — | 1 | 6.24 |
| CHEMBL1480783 | — | — | 1 | 6.23 |
| CHEMBL1964793 | — | — | 1 | 6.23 |
| CHEMBL1427476 | — | — | 1 | 6.23 |
| CHEMBL1314342 | — | — | 1 | 6.23 |
| CHEMBL1545088 | — | — | 1 | 6.21 |
| CHEMBL1448732 | — | — | 1 | 6.19 |
| CHEMBL3195591 | — | — | 1 | 6.19 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1313588 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL1543899 | — | IC50 | = | 260.0 | nM | 6.58 |
| CHEMBL1494293 | — | IC50 | = | 280.0 | nM | 6.55 |
| CHEMBL1339324 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL1340776 | — | IC50 | = | 330.0 | nM | 6.48 |
| CHEMBL508338 | THIMEROSAL | IC50 | = | 340.0 | nM | 6.47 |
| CHEMBL1562086 | — | IC50 | = | 340.0 | nM | 6.47 |
| CHEMBL1467760 | — | IC50 | = | 340.0 | nM | 6.47 |
| CHEMBL1417731 | — | IC50 | = | 360.0 | nM | 6.44 |
| CHEMBL1407492 | — | IC50 | = | 370.0 | nM | 6.43 |
| CHEMBL1335703 | — | IC50 | = | 370.0 | nM | 6.43 |
| CHEMBL1542899 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL1373411 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL1341756 | — | IC50 | = | 390.0 | nM | 6.41 |
| CHEMBL1303785 | — | IC50 | = | 430.0 | nM | 6.37 |
| CHEMBL1543127 | — | IC50 | = | 480.0 | nM | 6.32 |
| CHEMBL375781 | NEOCUPROINE | IC50 | = | 490.0 | nM | 6.31 |
| CHEMBL1396156 | — | IC50 | = | 490.0 | nM | 6.31 |
| CHEMBL1453396 | — | IC50 | = | 510.0 | nM | 6.29 |
| CHEMBL1556750 | — | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL1502870 | — | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL1420009 | — | IC50 | = | 540.0 | nM | 6.27 |
| CHEMBL1980982 | — | IC50 | = | 570.0 | nM | 6.24 |
| CHEMBL1480783 | — | IC50 | = | 590.0 | nM | 6.23 |
| CHEMBL1314342 | — | IC50 | = | 590.0 | nM | 6.23 |
| CHEMBL1964793 | — | IC50 | = | 590.0 | nM | 6.23 |
| CHEMBL1427476 | — | IC50 | = | 590.0 | nM | 6.23 |
| CHEMBL1545088 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL1448732 | — | IC50 | = | 650.0 | nM | 6.19 |
| CHEMBL3195591 | — | IC50 | = | 650.0 | nM | 6.19 |
| CHEMBL1522050 | — | IC50 | = | 660.0 | nM | 6.18 |
| CHEMBL1607882 | — | IC50 | = | 660.0 | nM | 6.18 |
| CHEMBL1373992 | — | IC50 | = | 660.0 | nM | 6.18 |
| CHEMBL1359688 | — | IC50 | = | 660.0 | nM | 6.18 |
| CHEMBL1472263 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL1535702 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL1415890 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL1433263 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL1597716 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL600060 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL1420768 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL478120 | MARBOFLOXACIN | IC50 | = | 720.0 | nM | 6.14 |
| CHEMBL1576407 | — | IC50 | = | 720.0 | nM | 6.14 |
| CHEMBL1378668 | — | IC50 | = | 730.0 | nM | 6.14 |
| CHEMBL1556481 | — | IC50 | = | 760.0 | nM | 6.12 |
| CHEMBL1524180 | — | IC50 | = | 750.0 | nM | 6.12 |
| CHEMBL3196253 | — | IC50 | = | 770.0 | nM | 6.11 |
| CHEMBL1476017 | — | IC50 | = | 780.0 | nM | 6.11 |
| CHEMBL1466340 | — | IC50 | = | 780.0 | nM | 6.11 |
| CHEMBL964 | DISULFIRAM | IC50 | = | 780.0 | nM | 6.11 |