Assay Detail
Functional
CHEMBL1614345
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response cell-based screening assay for antagonists of neuropeptide Y receptor Y2 (NPY-Y2). (Class of assay: confirmatory) [Related pubchem assays: 793, 1257, 1256 ]
119
Total Activities
119
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 119 | 5.19 | 6.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1543306 | — | — | 1 | 6.66 |
| CHEMBL1427860 | — | — | 1 | 6.53 |
| CHEMBL1398754 | — | — | 1 | 6.37 |
| CHEMBL1404069 | — | — | 1 | 6.13 |
| CHEMBL1353428 | — | — | 1 | 5.81 |
| CHEMBL1385608 | — | — | 1 | 5.78 |
| CHEMBL1585652 | — | — | 1 | 5.71 |
| CHEMBL1329549 | — | — | 1 | 5.53 |
| CHEMBL1428935 | — | — | 1 | 5.51 |
| CHEMBL1559259 | — | — | 1 | 5.50 |
| CHEMBL1439981 | — | — | 1 | 5.45 |
| CHEMBL3194054 | — | — | 1 | 5.45 |
| CHEMBL1608982 | — | — | 1 | 5.41 |
| CHEMBL3208997 | — | — | 1 | 5.38 |
| CHEMBL1423382 | — | — | 1 | 5.38 |
| CHEMBL417727 | — | — | 1 | 5.37 |
| CHEMBL1585445 | — | — | 1 | 5.37 |
| CHEMBL1468302 | — | — | 1 | 5.37 |
| CHEMBL1426022 | — | — | 1 | 5.36 |
| CHEMBL1312703 | — | — | 1 | 5.36 |
| CHEMBL1570844 | — | — | 1 | 5.36 |
| CHEMBL1365319 | — | — | 1 | 5.34 |
| CHEMBL3197426 | — | — | 1 | 5.34 |
| CHEMBL1487131 | — | — | 1 | 5.34 |
| CHEMBL262083 | N6-PHENYLADENOSINE | — | 1 | 5.33 |
| CHEMBL1493277 | — | — | 1 | 5.32 |
| CHEMBL1568243 | — | — | 1 | 5.30 |
| CHEMBL3190644 | — | — | 1 | 5.30 |
| CHEMBL1426896 | — | — | 1 | 5.30 |
| CHEMBL3211272 | — | — | 1 | 5.29 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1543306 | — | IC50 | = | 220.0 | nM | 6.66 |
| CHEMBL1427860 | — | IC50 | = | 298.0 | nM | 6.53 |
| CHEMBL1398754 | — | IC50 | = | 428.0 | nM | 6.37 |
| CHEMBL1404069 | — | IC50 | = | 733.0 | nM | 6.13 |
| CHEMBL1353428 | — | IC50 | = | 1564.0 | nM | 5.81 |
| CHEMBL1385608 | — | IC50 | = | 1647.0 | nM | 5.78 |
| CHEMBL1585652 | — | IC50 | = | 1974.0 | nM | 5.71 |
| CHEMBL1329549 | — | IC50 | = | 2949.0 | nM | 5.53 |
| CHEMBL1428935 | — | IC50 | = | 3064.0 | nM | 5.51 |
| CHEMBL1559259 | — | IC50 | = | 3137.0 | nM | 5.50 |
| CHEMBL3194054 | — | IC50 | = | 3550.0 | nM | 5.45 |
| CHEMBL1439981 | — | IC50 | = | 3546.0 | nM | 5.45 |
| CHEMBL1608982 | — | IC50 | = | 3917.0 | nM | 5.41 |
| CHEMBL1423382 | — | IC50 | = | 4120.0 | nM | 5.38 |
| CHEMBL3208997 | — | IC50 | = | 4180.0 | nM | 5.38 |
| CHEMBL417727 | — | IC50 | = | 4245.0 | nM | 5.37 |
| CHEMBL1585445 | — | IC50 | = | 4248.0 | nM | 5.37 |
| CHEMBL1468302 | — | IC50 | = | 4297.0 | nM | 5.37 |
| CHEMBL1570844 | — | IC50 | = | 4355.0 | nM | 5.36 |
| CHEMBL1312703 | — | IC50 | = | 4321.0 | nM | 5.36 |
| CHEMBL1426022 | — | IC50 | = | 4383.0 | nM | 5.36 |
| CHEMBL1487131 | — | IC50 | = | 4607.0 | nM | 5.34 |
| CHEMBL3197426 | — | IC50 | = | 4533.0 | nM | 5.34 |
| CHEMBL1365319 | — | IC50 | = | 4543.0 | nM | 5.34 |
| CHEMBL262083 | N6-PHENYLADENOSINE | IC50 | = | 4729.0 | nM | 5.33 |
| CHEMBL1493277 | — | IC50 | = | 4768.0 | nM | 5.32 |
| CHEMBL1568243 | — | IC50 | = | 4953.0 | nM | 5.30 |
| CHEMBL1426896 | — | IC50 | = | 5058.0 | nM | 5.30 |
| CHEMBL3190644 | — | IC50 | = | 4958.0 | nM | 5.30 |
| CHEMBL1599610 | — | IC50 | = | 5083.0 | nM | 5.29 |
| CHEMBL3211272 | — | IC50 | = | 5069.0 | nM | 5.29 |
| CHEMBL1308845 | — | IC50 | = | 5147.0 | nM | 5.29 |
| CHEMBL1389982 | — | IC50 | = | 5224.0 | nM | 5.28 |
| CHEMBL1427745 | — | IC50 | = | 5256.0 | nM | 5.28 |
| CHEMBL1423799 | — | IC50 | = | 5194.0 | nM | 5.28 |
| CHEMBL1499276 | — | IC50 | = | 5354.0 | nM | 5.27 |
| CHEMBL1345334 | — | IC50 | = | 5505.0 | nM | 5.26 |
| CHEMBL1402158 | — | IC50 | = | 5516.0 | nM | 5.26 |
| CHEMBL1431004 | — | IC50 | = | 5523.0 | nM | 5.26 |
| CHEMBL1308461 | — | IC50 | = | 5766.0 | nM | 5.24 |
| CHEMBL1468490 | — | IC50 | = | 5722.0 | nM | 5.24 |
| CHEMBL1545971 | — | IC50 | = | 5862.0 | nM | 5.23 |
| CHEMBL1360426 | — | IC50 | = | 6020.0 | nM | 5.22 |
| CHEMBL1427504 | — | IC50 | = | 6065.0 | nM | 5.22 |
| CHEMBL1366620 | — | IC50 | = | 6110.0 | nM | 5.21 |
| CHEMBL1432676 | — | IC50 | = | 6166.0 | nM | 5.21 |
| CHEMBL1574689 | — | IC50 | = | 6206.0 | nM | 5.21 |
| CHEMBL3214137 | — | IC50 | = | 6469.0 | nM | 5.19 |
| CHEMBL1531745 | — | IC50 | = | 6452.0 | nM | 5.19 |
| CHEMBL1522356 | — | IC50 | = | 6883.0 | nM | 5.16 |