Assay Detail
Functional
CHEMBL1614385
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Secondary Assay to Identify Inhibitors of Calcineurin. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1979, AID2007]
344
Total Activities
342
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Serine/threonine-protein phosphatase (CHEMBL1293271) ↗| Type | SINGLE PROTEIN |
| Organism | Candida dubliniensis (strain CD36 / CBS 7987 / NCPF 3949 / NRRLY-17841) (Yeast) |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 344 | 4.93 | 6.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1420556 | — | — | 1 | 6.08 |
| CHEMBL1546228 | — | — | 1 | 5.61 |
| CHEMBL3190873 | — | — | 1 | 5.59 |
| CHEMBL1386774 | — | — | 1 | 5.51 |
| CHEMBL1521297 | — | — | 1 | 5.42 |
| CHEMBL1328373 | — | — | 1 | 5.41 |
| CHEMBL1487639 | — | — | 1 | 5.41 |
| CHEMBL1469579 | — | — | 1 | 5.26 |
| CHEMBL1484777 | — | — | 1 | 5.09 |
| CHEMBL3198912 | — | — | 1 | 4.74 |
| CHEMBL1521991 | — | — | 1 | 4.74 |
| CHEMBL1596066 | — | — | 1 | 4.72 |
| CHEMBL1472105 | — | — | 1 | 4.69 |
| CHEMBL1382191 | — | — | 1 | 4.62 |
| CHEMBL1490555 | — | — | 1 | 4.61 |
| CHEMBL1514530 | — | — | 1 | 4.61 |
| CHEMBL1308052 | — | — | 1 | 4.55 |
| CHEMBL584442 | — | — | 1 | 4.53 |
| CHEMBL1502020 | — | — | 1 | 4.44 |
| CHEMBL601768 | — | — | 1 | 4.34 |
| CHEMBL1405204 | — | — | 1 | 4.34 |
| CHEMBL1587806 | — | — | 1 | 4.05 |
| CHEMBL600862 | — | — | 1 | - |
| CHEMBL1464485 | — | — | 1 | - |
| CHEMBL1477033 | — | — | 1 | - |
| CHEMBL1346226 | — | — | 1 | - |
| CHEMBL1319004 | — | — | 1 | - |
| CHEMBL1318943 | — | — | 1 | - |
| CHEMBL1408965 | — | — | 1 | - |
| CHEMBL1222385 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1420556 | — | EC50 | = | 828.0 | nM | 6.08 |
| CHEMBL1546228 | — | EC50 | = | 2468.0 | nM | 5.61 |
| CHEMBL3190873 | — | EC50 | = | 2578.0 | nM | 5.59 |
| CHEMBL1386774 | — | EC50 | = | 3074.0 | nM | 5.51 |
| CHEMBL1521297 | — | EC50 | = | 3784.0 | nM | 5.42 |
| CHEMBL1328373 | — | EC50 | = | 3921.0 | nM | 5.41 |
| CHEMBL1487639 | — | EC50 | = | 3925.0 | nM | 5.41 |
| CHEMBL1469579 | — | EC50 | = | 5548.0 | nM | 5.26 |
| CHEMBL1484777 | — | EC50 | = | 8099.0 | nM | 5.09 |
| CHEMBL3198912 | — | EC50 | = | 18232.0 | nM | 4.74 |
| CHEMBL1521991 | — | EC50 | = | 18149.0 | nM | 4.74 |
| CHEMBL1596066 | — | EC50 | = | 19245.0 | nM | 4.72 |
| CHEMBL1472105 | — | EC50 | = | 20218.0 | nM | 4.69 |
| CHEMBL1382191 | — | EC50 | = | 24159.0 | nM | 4.62 |
| CHEMBL1490555 | — | EC50 | = | 24723.0 | nM | 4.61 |
| CHEMBL1514530 | — | EC50 | = | 24836.0 | nM | 4.61 |
| CHEMBL1308052 | — | EC50 | = | 28074.0 | nM | 4.55 |
| CHEMBL584442 | — | EC50 | = | 29575.0 | nM | 4.53 |
| CHEMBL1502020 | — | EC50 | = | 36022.0 | nM | 4.44 |
| CHEMBL1405204 | — | EC50 | = | 45381.0 | nM | 4.34 |
| CHEMBL601768 | — | EC50 | = | 45383.0 | nM | 4.34 |
| CHEMBL1587806 | — | EC50 | = | 89128.0 | nM | 4.05 |
| CHEMBL1789993 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1373577 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1525081 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL602363 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1579999 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1351542 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1437579 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL3198836 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1524829 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1524956 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1570820 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1452090 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1462283 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1383916 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1609315 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1311007 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1383721 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1469362 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1383706 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1310713 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1979784 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1492378 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1485259 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1334557 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1350780 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL3196241 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL1548492 | — | EC50 | > | 180000.0 | nM | - |
| CHEMBL3145031 | — | EC50 | > | 180000.0 | nM | - |