Assay Detail
Binding
CHEMBL1614388
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: TR-FRET counterscreen for FAK inhibitors: dose-response biochemical high throughput screening assay to identify inhibitors of Proline-rich tyrosine kinase 2 (Pyk2). (Class of assay: confirmatory) [Related pubchem assays: 794, 727, 810 ]
211
Total Activities
210
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 211 | 5.23 | 6.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1384281 | — | — | 1 | 6.54 |
| CHEMBL255881 | — | — | 1 | 5.97 |
| CHEMBL1500600 | — | — | 1 | 5.91 |
| CHEMBL1323696 | — | — | 1 | 5.88 |
| CHEMBL1392806 | — | — | 1 | 5.84 |
| CHEMBL1345770 | — | — | 1 | 5.81 |
| CHEMBL1388603 | — | — | 2 | 5.80 |
| CHEMBL2002223 | — | — | 1 | 5.75 |
| CHEMBL1432963 | — | — | 1 | 5.74 |
| CHEMBL1347829 | — | — | 1 | 5.72 |
| CHEMBL1468746 | — | — | 1 | 5.72 |
| CHEMBL3192969 | — | — | 1 | 5.71 |
| CHEMBL1704267 | — | — | 1 | 5.70 |
| CHEMBL1370120 | — | — | 1 | 5.68 |
| CHEMBL1350854 | — | — | 1 | 5.67 |
| CHEMBL1351180 | — | — | 1 | 5.67 |
| CHEMBL1447467 | — | — | 1 | 5.67 |
| CHEMBL1577281 | — | — | 1 | 5.66 |
| CHEMBL1706577 | — | — | 1 | 5.65 |
| CHEMBL1414554 | — | — | 1 | 5.65 |
| CHEMBL1313195 | — | — | 1 | 5.64 |
| CHEMBL1346314 | — | — | 1 | 5.63 |
| CHEMBL374632 | — | — | 1 | 5.63 |
| CHEMBL1469742 | — | — | 1 | 5.61 |
| CHEMBL1349382 | — | — | 1 | 5.60 |
| CHEMBL1986591 | — | — | 1 | 5.59 |
| CHEMBL1380059 | — | — | 1 | 5.58 |
| CHEMBL1498729 | — | — | 1 | 5.58 |
| CHEMBL1714669 | — | — | 1 | 5.58 |
| CHEMBL1369422 | — | — | 1 | 5.57 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1384281 | — | IC50 | = | 288.0 | nM | 6.54 |
| CHEMBL255881 | — | IC50 | = | 1068.0 | nM | 5.97 |
| CHEMBL1500600 | — | IC50 | = | 1241.0 | nM | 5.91 |
| CHEMBL1323696 | — | IC50 | = | 1323.0 | nM | 5.88 |
| CHEMBL1392806 | — | IC50 | = | 1449.0 | nM | 5.84 |
| CHEMBL1345770 | — | IC50 | = | 1537.0 | nM | 5.81 |
| CHEMBL1388603 | — | IC50 | = | 1573.0 | nM | 5.80 |
| CHEMBL1388603 | — | IC50 | = | 1573.0 | nM | 5.80 |
| CHEMBL2002223 | — | IC50 | = | 1780.0 | nM | 5.75 |
| CHEMBL1432963 | — | IC50 | = | 1825.0 | nM | 5.74 |
| CHEMBL1468746 | — | IC50 | = | 1907.0 | nM | 5.72 |
| CHEMBL1347829 | — | IC50 | = | 1898.0 | nM | 5.72 |
| CHEMBL3192969 | — | IC50 | = | 1943.0 | nM | 5.71 |
| CHEMBL1704267 | — | IC50 | = | 2006.0 | nM | 5.70 |
| CHEMBL1370120 | — | IC50 | = | 2083.0 | nM | 5.68 |
| CHEMBL1350854 | — | IC50 | = | 2124.0 | nM | 5.67 |
| CHEMBL1351180 | — | IC50 | = | 2133.0 | nM | 5.67 |
| CHEMBL1447467 | — | IC50 | = | 2151.0 | nM | 5.67 |
| CHEMBL1577281 | — | IC50 | = | 2212.0 | nM | 5.66 |
| CHEMBL1414554 | — | IC50 | = | 2230.0 | nM | 5.65 |
| CHEMBL1706577 | — | IC50 | = | 2253.0 | nM | 5.65 |
| CHEMBL1313195 | — | IC50 | = | 2266.0 | nM | 5.64 |
| CHEMBL374632 | — | IC50 | = | 2324.0 | nM | 5.63 |
| CHEMBL1346314 | — | IC50 | = | 2368.0 | nM | 5.63 |
| CHEMBL1469742 | — | IC50 | = | 2444.0 | nM | 5.61 |
| CHEMBL1349382 | — | IC50 | = | 2498.0 | nM | 5.60 |
| CHEMBL1986591 | — | IC50 | = | 2567.0 | nM | 5.59 |
| CHEMBL1498729 | — | IC50 | = | 2660.0 | nM | 5.58 |
| CHEMBL1380059 | — | IC50 | = | 2637.0 | nM | 5.58 |
| CHEMBL1714669 | — | IC50 | = | 2647.0 | nM | 5.58 |
| CHEMBL1369422 | — | IC50 | = | 2704.0 | nM | 5.57 |
| CHEMBL1302158 | — | IC50 | = | 2718.0 | nM | 5.57 |
| CHEMBL341473 | — | IC50 | = | 2828.0 | nM | 5.55 |
| CHEMBL1574619 | — | IC50 | = | 2794.0 | nM | 5.55 |
| CHEMBL1334484 | — | IC50 | = | 2921.0 | nM | 5.53 |
| CHEMBL1467405 | — | IC50 | = | 3108.0 | nM | 5.51 |
| CHEMBL3197990 | — | IC50 | = | 3146.0 | nM | 5.50 |
| CHEMBL3199451 | — | IC50 | = | 3145.0 | nM | 5.50 |
| CHEMBL1492266 | — | IC50 | = | 3318.0 | nM | 5.48 |
| CHEMBL1327038 | — | IC50 | = | 3495.0 | nM | 5.46 |
| CHEMBL1542790 | — | IC50 | = | 3683.0 | nM | 5.43 |
| CHEMBL1456712 | — | IC50 | = | 3817.0 | nM | 5.42 |
| CHEMBL1482979 | — | IC50 | = | 3765.0 | nM | 5.42 |
| CHEMBL3189853 | — | IC50 | = | 3775.0 | nM | 5.42 |
| CHEMBL600336 | — | IC50 | = | 3974.0 | nM | 5.40 |
| CHEMBL1337717 | — | IC50 | = | 3989.0 | nM | 5.40 |
| CHEMBL1305250 | — | IC50 | = | 4085.0 | nM | 5.39 |
| CHEMBL1971613 | — | IC50 | = | 4307.0 | nM | 5.37 |
| CHEMBL1328311 | — | IC50 | = | 4281.0 | nM | 5.37 |
| CHEMBL1528600 | — | IC50 | = | 4254.0 | nM | 5.37 |