Assay Detail
Functional
CHEMBL1614390
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response assay for agonists of 5-Hydroxytryptamine (Serotonin) Receptor Subtype 1A (5HT1A). (Class of assay: confirmatory) [Related pubchem assays: 567, 574 ]
51
Total Activities
51
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 51 | 5.77 | 7.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1200791 | OXYMETAZOLINE HYDROCHLORIDE | 4.0 | 1 | 7.16 |
| CHEMBL1256400 | XYLOMETAZOLINE HYDROCHLORIDE | -1.0 | 1 | 6.89 |
| CHEMBL7257 | MEBUFOTENIN | 2.0 | 1 | 6.71 |
| CHEMBL1200938 | METHYSERGIDE MALEATE | 4.0 | 1 | 5.97 |
| CHEMBL1309229 | — | — | 1 | 5.74 |
| CHEMBL1507054 | — | — | 1 | 5.65 |
| CHEMBL348588 | — | — | 1 | 5.29 |
| CHEMBL26655 | — | — | 1 | 4.92 |
| CHEMBL1301276 | — | — | 1 | 4.86 |
| CHEMBL1523325 | — | — | 1 | 4.46 |
| CHEMBL1373172 | — | — | 1 | - |
| CHEMBL1588802 | — | — | 1 | - |
| CHEMBL1492495 | — | — | 1 | - |
| CHEMBL27811 | — | — | 1 | - |
| CHEMBL1511639 | — | — | 1 | - |
| CHEMBL1334769 | — | — | 1 | - |
| CHEMBL1550957 | — | — | 1 | - |
| CHEMBL1492488 | — | — | 1 | - |
| CHEMBL1328749 | — | — | 1 | - |
| CHEMBL3199532 | — | — | 1 | - |
| CHEMBL1452784 | — | — | 1 | - |
| CHEMBL587229 | — | — | 1 | - |
| CHEMBL1548144 | — | — | 1 | - |
| CHEMBL1310557 | — | — | 1 | - |
| CHEMBL1428589 | — | — | 1 | - |
| CHEMBL1456789 | — | — | 1 | - |
| CHEMBL1477013 | — | — | 1 | - |
| CHEMBL1377426 | — | — | 1 | - |
| CHEMBL1494440 | — | — | 1 | - |
| CHEMBL1455750 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1200791 | OXYMETAZOLINE HYDROCHLORIDE | EC50 | = | 70.0 | nM | 7.16 |
| CHEMBL1256400 | XYLOMETAZOLINE HYDROCHLORIDE | EC50 | = | 129.0 | nM | 6.89 |
| CHEMBL7257 | MEBUFOTENIN | EC50 | = | 197.0 | nM | 6.71 |
| CHEMBL1200938 | METHYSERGIDE MALEATE | EC50 | = | 1075.0 | nM | 5.97 |
| CHEMBL1309229 | — | EC50 | = | 1815.0 | nM | 5.74 |
| CHEMBL1507054 | — | EC50 | = | 2219.0 | nM | 5.65 |
| CHEMBL348588 | — | EC50 | = | 5100.0 | nM | 5.29 |
| CHEMBL26655 | — | EC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL1301276 | — | EC50 | = | 13800.0 | nM | 4.86 |
| CHEMBL1523325 | — | EC50 | = | 34800.0 | nM | 4.46 |
| CHEMBL1527675 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL3196650 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1409828 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL544428 | MIANSERIN HYDROCHLORIDE | EC50 | > | 50000.0 | nM | - |
| CHEMBL1361184 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1578139 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1381546 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1595470 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1438062 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1410188 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1465394 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1559501 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1375660 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1463453 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1345618 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1464351 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1542860 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1454839 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1606397 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1528874 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1452784 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1455750 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1494440 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1377426 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1477013 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1456789 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1428589 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1310557 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1548144 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL587229 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL3199532 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1373172 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1588802 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1492495 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL27811 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1511639 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1334769 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1550957 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1492488 | — | EC50 | > | 50000.0 | nM | - |
| CHEMBL1328749 | — | EC50 | > | 50000.0 | nM | - |