Assay Detail
Functional
CHEMBL1614407
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence-based counterscreen for agonists of NPY-Y2: cell-based high-throughput dose response assay for agonists of NPY-Y1. (Class of assay: confirmatory) [Related pubchem assays: 1703 (Screening assay (CNGC inhibitors).), 1359 (Screening assay (NPY-Y2 potentiators or agonists).), 1304 (Screening assay (NPY-Y1 potentiators or agonists).), 1710 (Screening assay (NPY-Y2 agonists).), 1791 (Summary AID.)]
89
Total Activities
89
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 89 | 4.87 | 5.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1454903 | — | — | 1 | 5.51 |
| CHEMBL1549309 | — | — | 1 | 5.47 |
| CHEMBL1311742 | — | — | 1 | 5.22 |
| CHEMBL1519263 | — | — | 1 | 5.19 |
| CHEMBL1373205 | — | — | 1 | 5.18 |
| CHEMBL1573719 | — | — | 1 | 5.15 |
| CHEMBL1374954 | — | — | 1 | 5.13 |
| CHEMBL1366987 | — | — | 1 | 5.09 |
| CHEMBL1548605 | — | — | 1 | 5.07 |
| CHEMBL3194195 | — | — | 1 | 5.03 |
| CHEMBL1342462 | — | — | 1 | 5.02 |
| CHEMBL2062335 | METOPROLOL TARTRATE | 4.0 | 1 | 5.02 |
| CHEMBL496 | HEXACHLOROPHENE | 4.0 | 1 | 5.01 |
| CHEMBL1471202 | — | — | 1 | 5.00 |
| CHEMBL3213459 | — | — | 1 | 4.97 |
| CHEMBL1322039 | — | — | 1 | 4.96 |
| CHEMBL1547757 | — | — | 1 | 4.94 |
| CHEMBL1581332 | — | — | 1 | 4.93 |
| CHEMBL3213319 | — | — | 1 | 4.91 |
| CHEMBL1482637 | — | — | 1 | 4.90 |
| CHEMBL1299267 | — | — | 1 | 4.90 |
| CHEMBL1602800 | — | — | 1 | 4.89 |
| CHEMBL1329027 | — | — | 1 | 4.88 |
| CHEMBL1505552 | — | — | 1 | 4.83 |
| CHEMBL1583097 | — | — | 1 | 4.80 |
| CHEMBL1431189 | — | — | 1 | 4.78 |
| CHEMBL1309183 | — | — | 1 | 4.78 |
| CHEMBL3192204 | — | — | 1 | 4.78 |
| CHEMBL1544847 | — | — | 1 | 4.77 |
| CHEMBL1378687 | — | — | 1 | 4.76 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1454903 | — | EC50 | = | 3068.0 | nM | 5.51 |
| CHEMBL1549309 | — | EC50 | = | 3408.0 | nM | 5.47 |
| CHEMBL1311742 | — | EC50 | = | 5996.0 | nM | 5.22 |
| CHEMBL1519263 | — | EC50 | = | 6462.0 | nM | 5.19 |
| CHEMBL1373205 | — | EC50 | = | 6636.0 | nM | 5.18 |
| CHEMBL1573719 | — | EC50 | = | 7053.0 | nM | 5.15 |
| CHEMBL1374954 | — | EC50 | = | 7410.0 | nM | 5.13 |
| CHEMBL1366987 | — | EC50 | = | 8195.0 | nM | 5.09 |
| CHEMBL1548605 | — | EC50 | = | 8504.0 | nM | 5.07 |
| CHEMBL3194195 | — | EC50 | = | 9377.0 | nM | 5.03 |
| CHEMBL1342462 | — | EC50 | = | 9489.0 | nM | 5.02 |
| CHEMBL2062335 | METOPROLOL TARTRATE | EC50 | = | 9606.0 | nM | 5.02 |
| CHEMBL496 | HEXACHLOROPHENE | EC50 | = | 9796.0 | nM | 5.01 |
| CHEMBL1471202 | — | EC50 | = | 9924.0 | nM | 5.00 |
| CHEMBL3213459 | — | EC50 | = | 10621.0 | nM | 4.97 |
| CHEMBL1322039 | — | EC50 | = | 10864.0 | nM | 4.96 |
| CHEMBL1547757 | — | EC50 | = | 11573.0 | nM | 4.94 |
| CHEMBL1581332 | — | EC50 | = | 11701.0 | nM | 4.93 |
| CHEMBL3213319 | — | EC50 | = | 12355.0 | nM | 4.91 |
| CHEMBL1482637 | — | EC50 | = | 12619.0 | nM | 4.90 |
| CHEMBL1299267 | — | EC50 | = | 12496.0 | nM | 4.90 |
| CHEMBL1602800 | — | EC50 | = | 12746.0 | nM | 4.89 |
| CHEMBL1329027 | — | EC50 | = | 13279.0 | nM | 4.88 |
| CHEMBL1505552 | — | EC50 | = | 14783.0 | nM | 4.83 |
| CHEMBL1583097 | — | EC50 | = | 15697.0 | nM | 4.80 |
| CHEMBL1431189 | — | EC50 | = | 16500.0 | nM | 4.78 |
| CHEMBL3192204 | — | EC50 | = | 16470.0 | nM | 4.78 |
| CHEMBL1309183 | — | EC50 | = | 16732.0 | nM | 4.78 |
| CHEMBL1544847 | — | EC50 | = | 17105.0 | nM | 4.77 |
| CHEMBL1378687 | — | EC50 | = | 17280.0 | nM | 4.76 |
| CHEMBL1541596 | — | EC50 | = | 18547.0 | nM | 4.73 |
| CHEMBL1431891 | — | EC50 | = | 18569.0 | nM | 4.73 |
| CHEMBL1537587 | — | EC50 | = | 19303.0 | nM | 4.71 |
| CHEMBL1345141 | — | EC50 | = | 22043.0 | nM | 4.66 |
| CHEMBL1538646 | — | EC50 | = | 21818.0 | nM | 4.66 |
| CHEMBL1517881 | — | EC50 | = | 22163.0 | nM | 4.65 |
| CHEMBL1343823 | — | EC50 | = | 24380.0 | nM | 4.61 |
| CHEMBL1302519 | — | EC50 | = | 24391.0 | nM | 4.61 |
| CHEMBL1392858 | — | EC50 | = | 26411.0 | nM | 4.58 |
| CHEMBL1418821 | — | EC50 | = | 26506.0 | nM | 4.58 |
| CHEMBL1447448 | — | EC50 | = | 28902.0 | nM | 4.54 |
| CHEMBL1995800 | — | EC50 | = | 33309.0 | nM | 4.48 |
| CHEMBL1336098 | — | EC50 | = | 33757.0 | nM | 4.47 |
| CHEMBL1504701 | — | EC50 | = | 35337.0 | nM | 4.45 |
| CHEMBL2004475 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1388940 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL3197361 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1428620 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL3198532 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1350193 | — | EC50 | > | 35430.0 | nM | - |