Assay Detail
Functional
CHEMBL1614467
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Late stage fluorescence dose response cell-based screening assay for antagonists of the Sphingosine 1-Phosphate Receptor 4 (S1P4). (Class of assay: confirmatory) [Related pubchem assays: 1524 (Confirmation screen (S1P4 antagonists).), 1510 (Primary screen (S1P4 antagonists).), 1853 (Summary AID (S1P4 antagonists).), 1692 (Dose response screen (S1P4 antagonists).)]
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 29 | 5.64 | 7.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1415555 | — | — | 1 | 7.41 |
| CHEMBL1603615 | — | — | 1 | 7.08 |
| CHEMBL1412583 | — | — | 1 | 6.47 |
| CHEMBL1331049 | — | — | 1 | 6.47 |
| CHEMBL1487635 | — | — | 1 | 6.26 |
| CHEMBL1369594 | — | — | 1 | 6.13 |
| CHEMBL1390139 | — | — | 1 | 6.11 |
| CHEMBL1362503 | — | — | 1 | 6.05 |
| CHEMBL1439384 | — | — | 1 | 5.94 |
| CHEMBL213580 | — | — | 1 | 5.85 |
| CHEMBL1413680 | — | — | 1 | 5.76 |
| CHEMBL1446971 | — | — | 1 | 5.74 |
| CHEMBL1341981 | — | — | 1 | 5.54 |
| CHEMBL1449794 | — | — | 1 | 5.46 |
| CHEMBL1370681 | — | — | 1 | 5.46 |
| CHEMBL1429929 | — | — | 1 | 5.45 |
| CHEMBL1529115 | — | — | 1 | 5.43 |
| CHEMBL1569585 | — | — | 1 | 5.43 |
| CHEMBL1486934 | — | — | 1 | 5.35 |
| CHEMBL1502358 | — | — | 1 | 5.34 |
| CHEMBL1369655 | — | — | 1 | 5.28 |
| CHEMBL1299526 | — | — | 1 | 5.17 |
| CHEMBL1450393 | — | — | 1 | 5.01 |
| CHEMBL1543295 | — | — | 1 | 4.97 |
| CHEMBL1333510 | — | — | 1 | 4.95 |
| CHEMBL1424562 | — | — | 1 | 4.92 |
| CHEMBL1309232 | — | — | 1 | 4.81 |
| CHEMBL1334984 | — | — | 1 | 4.05 |
| CHEMBL1451470 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1415555 | — | IC50 | = | 39.27 | nM | 7.41 |
| CHEMBL1603615 | — | IC50 | = | 82.66 | nM | 7.08 |
| CHEMBL1412583 | — | IC50 | = | 342.1 | nM | 6.47 |
| CHEMBL1331049 | — | IC50 | = | 338.5 | nM | 6.47 |
| CHEMBL1487635 | — | IC50 | = | 550.2 | nM | 6.26 |
| CHEMBL1369594 | — | IC50 | = | 737.5 | nM | 6.13 |
| CHEMBL1390139 | — | IC50 | = | 770.3 | nM | 6.11 |
| CHEMBL1362503 | — | IC50 | = | 886.7 | nM | 6.05 |
| CHEMBL1439384 | — | IC50 | = | 1149.0 | nM | 5.94 |
| CHEMBL213580 | — | IC50 | = | 1423.0 | nM | 5.85 |
| CHEMBL1413680 | — | IC50 | = | 1723.0 | nM | 5.76 |
| CHEMBL1446971 | — | IC50 | = | 1804.0 | nM | 5.74 |
| CHEMBL1341981 | — | IC50 | = | 2894.0 | nM | 5.54 |
| CHEMBL1449794 | — | IC50 | = | 3493.0 | nM | 5.46 |
| CHEMBL1370681 | — | IC50 | = | 3453.0 | nM | 5.46 |
| CHEMBL1429929 | — | IC50 | = | 3584.0 | nM | 5.45 |
| CHEMBL1529115 | — | IC50 | = | 3715.0 | nM | 5.43 |
| CHEMBL1569585 | — | IC50 | = | 3697.0 | nM | 5.43 |
| CHEMBL1486934 | — | IC50 | = | 4510.0 | nM | 5.35 |
| CHEMBL1502358 | — | IC50 | = | 4548.0 | nM | 5.34 |
| CHEMBL1369655 | — | IC50 | = | 5278.0 | nM | 5.28 |
| CHEMBL1299526 | — | IC50 | = | 6739.0 | nM | 5.17 |
| CHEMBL1450393 | — | IC50 | = | 9683.0 | nM | 5.01 |
| CHEMBL1543295 | — | IC50 | = | 10760.0 | nM | 4.97 |
| CHEMBL1333510 | — | IC50 | = | 11210.0 | nM | 4.95 |
| CHEMBL1424562 | — | IC50 | = | 12020.0 | nM | 4.92 |
| CHEMBL1309232 | — | IC50 | = | 15430.0 | nM | 4.81 |
| CHEMBL1334984 | — | IC50 | = | 88820.0 | nM | 4.05 |
| CHEMBL1451470 | — | IC50 | > | 50000.0 | nM | - |