Assay Detail
Functional
CHEMBL1614475
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Cytotoxicity assay in HEK293 cells. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1266, AID1269, AID1270, AID1271, AID1280, AID1281, AID1282, AID1283, AID1287, AID1289, AID1290, AID1291, AID1292, AID1293, AID1294, AID1295, AID1299, AID1302, AID1364, AID1365, AID1366, AID1367, AID1369, AID1370, AID1371, AID1372, AID1373, AID1374, AID1375, AID1384, AID465]
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 27 | 5.11 | 6.23 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1372889 | — | — | 1 | 6.23 |
| CHEMBL1482541 | — | — | 1 | 5.66 |
| CHEMBL1401969 | — | — | 1 | 5.24 |
| CHEMBL1370087 | — | — | 1 | 5.09 |
| CHEMBL1170624 | — | — | 1 | 5.07 |
| CHEMBL1504484 | — | — | 1 | 4.99 |
| CHEMBL42529 | — | — | 1 | 4.91 |
| CHEMBL1518672 | — | — | 1 | 4.88 |
| CHEMBL1566033 | — | — | 1 | 4.86 |
| CHEMBL1576870 | — | — | 1 | 4.83 |
| CHEMBL1172202 | — | — | 1 | 4.81 |
| CHEMBL1578584 | — | — | 1 | 4.69 |
| CHEMBL1589625 | — | — | 1 | - |
| CHEMBL1611128 | — | — | 1 | - |
| CHEMBL373137 | — | — | 1 | - |
| CHEMBL1427791 | — | — | 1 | - |
| CHEMBL1600399 | — | — | 1 | - |
| CHEMBL1403324 | — | — | 1 | - |
| CHEMBL1410454 | — | — | 1 | - |
| CHEMBL1407693 | — | — | 1 | - |
| CHEMBL1491842 | — | — | 1 | - |
| CHEMBL1579418 | — | — | 1 | - |
| CHEMBL363657 | — | — | 1 | - |
| CHEMBL1557774 | — | — | 1 | - |
| CHEMBL1309478 | — | — | 1 | - |
| CHEMBL1410813 | — | — | 1 | - |
| CHEMBL1579491 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1372889 | — | EC50 | = | 588.6 | nM | 6.23 |
| CHEMBL1482541 | — | EC50 | = | 2192.0 | nM | 5.66 |
| CHEMBL1401969 | — | EC50 | = | 5717.0 | nM | 5.24 |
| CHEMBL1370087 | — | EC50 | = | 8144.0 | nM | 5.09 |
| CHEMBL1170624 | — | EC50 | = | 8481.0 | nM | 5.07 |
| CHEMBL1504484 | — | EC50 | = | 10220.0 | nM | 4.99 |
| CHEMBL42529 | — | EC50 | = | 12200.0 | nM | 4.91 |
| CHEMBL1518672 | — | EC50 | = | 13090.0 | nM | 4.88 |
| CHEMBL1566033 | — | EC50 | = | 13900.0 | nM | 4.86 |
| CHEMBL1576870 | — | EC50 | = | 14940.0 | nM | 4.83 |
| CHEMBL1172202 | — | EC50 | = | 15480.0 | nM | 4.81 |
| CHEMBL1578584 | — | EC50 | = | 20320.0 | nM | 4.69 |
| CHEMBL1589625 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1611128 | — | EC50 | > | 13250.0 | nM | - |
| CHEMBL373137 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1427791 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1600399 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1403324 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1410454 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1407693 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1491842 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1579418 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL363657 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1557774 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1309478 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1410813 | — | EC50 | > | 8000.0 | nM | - |
| CHEMBL1579491 | — | EC50 | > | 8000.0 | nM | - |