Assay Detail
Functional
CHEMBL1614514
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescent assay for HTS discovery of chemical activators of placental alkaline phosphatase. (Class of assay: confirmatory) [Related pubchem assays: 518 ]
254
Total Activities
254
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Alkaline phosphatase, germ cell type (CHEMBL3402) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 254 | 4.58 | 6.69 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1302272 | — | — | 1 | 6.69 |
| CHEMBL1336276 | — | — | 1 | 6.34 |
| CHEMBL1302946 | — | — | 1 | 5.96 |
| CHEMBL1572262 | — | — | 1 | 5.58 |
| CHEMBL1459455 | — | — | 1 | 5.48 |
| CHEMBL1599901 | — | — | 1 | 5.10 |
| CHEMBL1579513 | — | — | 1 | 5.07 |
| CHEMBL1403606 | — | — | 1 | 5.04 |
| CHEMBL1976754 | — | — | 1 | 4.96 |
| CHEMBL1458324 | — | — | 1 | 4.75 |
| CHEMBL1409782 | — | — | 1 | 4.68 |
| CHEMBL1428640 | — | — | 1 | 4.67 |
| CHEMBL1454476 | — | — | 1 | 4.64 |
| CHEMBL1495555 | — | — | 1 | 4.63 |
| CHEMBL1379607 | — | — | 1 | 4.61 |
| CHEMBL610508 | — | — | 1 | 4.60 |
| CHEMBL1325006 | — | — | 1 | 4.59 |
| CHEMBL1462208 | — | — | 1 | 4.58 |
| CHEMBL1559056 | — | — | 1 | 4.45 |
| CHEMBL1392552 | — | — | 1 | 4.43 |
| CHEMBL1988579 | — | — | 1 | 4.42 |
| CHEMBL1412954 | — | — | 1 | 4.41 |
| CHEMBL1991234 | — | — | 1 | 4.32 |
| CHEMBL1311641 | — | — | 1 | 4.31 |
| CHEMBL1594922 | — | — | 1 | 4.29 |
| CHEMBL3198436 | — | — | 1 | 4.26 |
| CHEMBL3198168 | — | — | 1 | 4.23 |
| CHEMBL1605701 | — | — | 1 | 4.21 |
| CHEMBL1407614 | — | — | 1 | 4.20 |
| CHEMBL1516984 | — | — | 1 | 4.18 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1302272 | — | EC50 | = | 203.0 | nM | 6.69 |
| CHEMBL1336276 | — | EC50 | = | 457.0 | nM | 6.34 |
| CHEMBL1302946 | — | EC50 | = | 1090.0 | nM | 5.96 |
| CHEMBL1572262 | — | EC50 | = | 2650.0 | nM | 5.58 |
| CHEMBL1459455 | — | EC50 | = | 3310.0 | nM | 5.48 |
| CHEMBL1599901 | — | EC50 | = | 7890.0 | nM | 5.10 |
| CHEMBL1579513 | — | EC50 | = | 8520.0 | nM | 5.07 |
| CHEMBL1403606 | — | EC50 | = | 9080.0 | nM | 5.04 |
| CHEMBL1976754 | — | EC50 | = | 10900.0 | nM | 4.96 |
| CHEMBL1458324 | — | EC50 | = | 17700.0 | nM | 4.75 |
| CHEMBL1409782 | — | EC50 | = | 21100.0 | nM | 4.68 |
| CHEMBL1428640 | — | EC50 | = | 21400.0 | nM | 4.67 |
| CHEMBL1454476 | — | EC50 | = | 23100.0 | nM | 4.64 |
| CHEMBL1495555 | — | EC50 | = | 23400.0 | nM | 4.63 |
| CHEMBL1379607 | — | EC50 | = | 24800.0 | nM | 4.61 |
| CHEMBL610508 | — | EC50 | = | 25300.0 | nM | 4.60 |
| CHEMBL1325006 | — | EC50 | = | 25900.0 | nM | 4.59 |
| CHEMBL1462208 | — | EC50 | = | 26300.0 | nM | 4.58 |
| CHEMBL1559056 | — | EC50 | = | 35600.0 | nM | 4.45 |
| CHEMBL1392552 | — | EC50 | = | 37000.0 | nM | 4.43 |
| CHEMBL1988579 | — | EC50 | = | 38400.0 | nM | 4.42 |
| CHEMBL1412954 | — | EC50 | = | 39200.0 | nM | 4.41 |
| CHEMBL1991234 | — | EC50 | = | 48200.0 | nM | 4.32 |
| CHEMBL1311641 | — | EC50 | = | 48500.0 | nM | 4.31 |
| CHEMBL1594922 | — | EC50 | = | 51000.0 | nM | 4.29 |
| CHEMBL3198436 | — | EC50 | = | 54500.0 | nM | 4.26 |
| CHEMBL3198168 | — | EC50 | = | 59200.0 | nM | 4.23 |
| CHEMBL1605701 | — | EC50 | = | 61900.0 | nM | 4.21 |
| CHEMBL1407614 | — | EC50 | = | 63100.0 | nM | 4.20 |
| CHEMBL1516984 | — | EC50 | = | 66500.0 | nM | 4.18 |
| CHEMBL1532795 | — | EC50 | = | 65900.0 | nM | 4.18 |
| CHEMBL1499077 | — | EC50 | = | 66900.0 | nM | 4.17 |
| CHEMBL1400955 | — | EC50 | = | 69400.0 | nM | 4.16 |
| CHEMBL3193915 | — | EC50 | = | 72100.0 | nM | 4.14 |
| CHEMBL1584202 | — | EC50 | = | 74000.0 | nM | 4.13 |
| CHEMBL1495574 | — | EC50 | = | 78000.0 | nM | 4.11 |
| CHEMBL1340701 | — | EC50 | = | 78500.0 | nM | 4.11 |
| CHEMBL1303708 | — | EC50 | = | 77200.0 | nM | 4.11 |
| CHEMBL1334710 | — | EC50 | = | 79400.0 | nM | 4.10 |
| CHEMBL1439775 | — | EC50 | = | 82800.0 | nM | 4.08 |
| CHEMBL1527041 | — | EC50 | = | 86800.0 | nM | 4.06 |
| CHEMBL1601093 | — | EC50 | = | 94100.0 | nM | 4.03 |
| CHEMBL1385608 | — | EC50 | = | 99600.0 | nM | 4.00 |
| CHEMBL1365415 | — | EC50 | = | 999000.0 | nM | - |
| CHEMBL1404792 | — | EC50 | = | 999000.0 | nM | - |
| CHEMBL1534915 | — | EC50 | = | 999000.0 | nM | - |
| CHEMBL1506480 | — | EC50 | = | 999000.0 | nM | - |
| CHEMBL1388509 | — | EC50 | = | 999000.0 | nM | - |
| CHEMBL1506384 | — | EC50 | = | 999000.0 | nM | - |
| CHEMBL1496045 | — | EC50 | = | 999000.0 | nM | - |