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Compound Detail

CHEMBL1302946

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Cc1cccc(N2C(=O)NC(=O)/C(=C\c3cnn(-c4ccccc4)c3)C2=O)c1

Basic Information

ChEMBL ID CHEMBL1302946
Phase Preclinical
Structure Type MOL
InChI Key IZYLJRRYKPUHJW-WOJGMQOQSA-N
2
Targets
3
Activities
2
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

372.4
MW (Da)
2.85
ALogP
5
HBA
1
HBD
84.3
PSA (Ų)
0.57
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C21H16N4O3
MW 372.38
Aromatic Rings 3
Heavy Atoms 28
NP-Likeness -1.90

Activity Summary

EC50 2 meas. best 5.96
IC50 1 meas.

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Alkaline phosphatase, germ cell type
CHEMBL3402
EC50 5.96 5.96 1090.0 1
Neurotensin receptor type 1
CHEMBL4123
EC50 4.89 4.89 13000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine