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Compound Detail

CHEMBL3193915

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Cc1nn(C)cc1/C=N\NC(=O)c1ccc2c(c1)c(C)c(C)n2Cc1ccccc1

Basic Information

ChEMBL ID CHEMBL3193915
Phase Preclinical
Structure Type MOL
InChI Key XATNJMFESTVZDB-MXAYSNPKSA-N
2
Targets
3
Activities
2
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

399.5
MW (Da)
4.11
ALogP
5
HBA
1
HBD
64.2
PSA (Ų)
0.41
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C24H25N5O
MW 399.50
Aromatic Rings 4
Heavy Atoms 30
NP-Likeness -2.02

Activity Summary

EC50 2 meas. best 4.17
IC50 1 meas.

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Heat shock factor protein 1
CHEMBL5313
EC50 4.17 4.17 67680.0 1
Alkaline phosphatase, germ cell type
CHEMBL3402
EC50 4.14 4.14 72100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine