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Assay Detail

CHEMBL1676508

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Functional
Antifungal activity against 5 x 10'6 CFU/ml Trichophyton quinckeanum B68683 by resazurin based fluorimetry assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Trichophyton quinckeanum
Confidence 1 — Organism
Curated By Autocuration

Target

Trichophyton quinckeanum (CHEMBL612334)
Type ORGANISM
Organism Trichophyton quinckeanum

Publication

In vitro profiling of pramiconazole and in vivo evaluation in Microsporum canis dermatitis and Candida albicans vaginitis laboratory models.
de Wit K, Paulussen C, Matheeussen A, van Rossem K, Cos P, Maes L.
Antimicrob Agents Chemother (2010) 54 : 4927 -4929
PubMed 20805398 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 6.38 8.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL822 TERBINAFINE 4.0 1 8.00
CHEMBL91 MICONAZOLE 4.0 1 6.10
CHEMBL175633 PRAMICONAZOLE 2.0 1 5.87
CHEMBL64391 ITRACONAZOLE 4.0 1 5.53

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL822 TERBINAFINE IC50 = 10.0 nM 8.00
CHEMBL91 MICONAZOLE IC50 = 790.0 nM 6.10
CHEMBL175633 PRAMICONAZOLE IC50 = 1340.0 nM 5.87
CHEMBL64391 ITRACONAZOLE IC50 = 2930.0 nM 5.53