Assay Detail
Functional
CHEMBL1737900
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR LYP1 Fluorescent Assay using pCAP substrate for In Vitro dose response studies - Set 2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1779, AID1784, AID2135, AID449727]
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Tyrosine-protein phosphatase non-receptor type 22 (CHEMBL2889) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 34 | 5.11 | 6.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1701224 | — | — | 1 | 6.60 |
| CHEMBL1438889 | — | — | 1 | 5.86 |
| CHEMBL1443268 | — | — | 1 | 5.80 |
| CHEMBL1320181 | — | — | 1 | 5.73 |
| CHEMBL1492305 | — | — | 1 | 5.51 |
| CHEMBL1439815 | — | — | 1 | 5.50 |
| CHEMBL1390354 | — | — | 1 | 5.46 |
| CHEMBL1704862 | — | — | 1 | 5.43 |
| CHEMBL1719149 | — | — | 1 | 5.39 |
| CHEMBL1456664 | — | — | 1 | 5.36 |
| CHEMBL1572439 | — | — | 1 | 5.26 |
| CHEMBL1371816 | — | — | 1 | 5.18 |
| CHEMBL1550429 | — | — | 1 | 5.16 |
| CHEMBL1724482 | — | — | 1 | 4.97 |
| CHEMBL1722719 | — | — | 1 | 4.91 |
| CHEMBL1562411 | — | — | 1 | 4.66 |
| CHEMBL1706168 | — | — | 1 | 4.47 |
| CHEMBL1718018 | — | — | 1 | 4.44 |
| CHEMBL1417070 | — | — | 1 | 4.35 |
| CHEMBL1729772 | — | — | 1 | 4.26 |
| CHEMBL1425801 | — | — | 1 | 4.09 |
| CHEMBL1714966 | — | — | 1 | 4.06 |
| CHEMBL1713374 | — | — | 1 | - |
| CHEMBL1732934 | — | — | 1 | - |
| CHEMBL1721448 | — | — | 1 | - |
| CHEMBL1400747 | — | — | 1 | - |
| CHEMBL1710376 | — | — | 1 | - |
| CHEMBL1700415 | — | — | 1 | - |
| CHEMBL1715912 | — | — | 1 | - |
| CHEMBL1488869 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1701224 | — | IC50 | = | 249.0 | nM | 6.60 |
| CHEMBL1438889 | — | IC50 | = | 1380.0 | nM | 5.86 |
| CHEMBL1443268 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL1320181 | — | IC50 | = | 1860.0 | nM | 5.73 |
| CHEMBL1492305 | — | IC50 | = | 3100.0 | nM | 5.51 |
| CHEMBL1439815 | — | IC50 | = | 3170.0 | nM | 5.50 |
| CHEMBL1390354 | — | IC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL1704862 | — | IC50 | = | 3680.0 | nM | 5.43 |
| CHEMBL1719149 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL1456664 | — | IC50 | = | 4420.0 | nM | 5.36 |
| CHEMBL1572439 | — | IC50 | = | 5520.0 | nM | 5.26 |
| CHEMBL1371816 | — | IC50 | = | 6540.0 | nM | 5.18 |
| CHEMBL1550429 | — | IC50 | = | 6890.0 | nM | 5.16 |
| CHEMBL1724482 | — | IC50 | = | 10800.0 | nM | 4.97 |
| CHEMBL1722719 | — | IC50 | = | 12200.0 | nM | 4.91 |
| CHEMBL1562411 | — | IC50 | = | 22100.0 | nM | 4.66 |
| CHEMBL1706168 | — | IC50 | = | 33900.0 | nM | 4.47 |
| CHEMBL1718018 | — | IC50 | = | 36100.0 | nM | 4.44 |
| CHEMBL1417070 | — | IC50 | = | 45000.0 | nM | 4.35 |
| CHEMBL1729772 | — | IC50 | = | 55000.0 | nM | 4.26 |
| CHEMBL1425801 | — | IC50 | = | 81200.0 | nM | 4.09 |
| CHEMBL1714966 | — | IC50 | = | 86700.0 | nM | 4.06 |
| CHEMBL1713374 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1732934 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1721448 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1400747 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1710376 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1700415 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1715912 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1488869 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1719458 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1735637 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1461397 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1478943 | — | IC50 | > | 100000.0 | nM | - |