Assay Detail
Functional
CHEMBL1738131
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response selectivity of uHTS chemical inhibitors of B-cell specific antigen receptor-induced NF-kB activation in Jurkat cells using a luminescence assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID435022, AID435025, AID465]
470
Total Activities
469
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | Jurkat |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 470 | 5.11 | 6.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1350077 | — | — | 1 | 6.75 |
| CHEMBL1965654 | — | — | 1 | 6.68 |
| CHEMBL1300766 | — | — | 1 | 6.66 |
| CHEMBL1559811 | — | — | 1 | 6.64 |
| CHEMBL1528660 | — | — | 1 | 6.62 |
| CHEMBL1305304 | — | — | 1 | 6.60 |
| CHEMBL1320514 | — | — | 1 | 6.58 |
| CHEMBL1505655 | — | — | 1 | 6.48 |
| CHEMBL1352270 | — | — | 1 | 6.48 |
| CHEMBL1484661 | — | — | 1 | 6.47 |
| CHEMBL1418371 | — | — | 1 | 6.44 |
| CHEMBL1521793 | — | — | 1 | 6.41 |
| CHEMBL1302818 | — | — | 1 | 6.40 |
| CHEMBL1369231 | — | — | 1 | 6.34 |
| CHEMBL1351755 | — | — | 1 | 6.33 |
| CHEMBL1393156 | — | — | 1 | 6.28 |
| CHEMBL1465119 | — | — | 1 | 6.24 |
| CHEMBL1255937 | ANCITABINE HYDROCHLORIDE | — | 1 | 6.19 |
| CHEMBL1430068 | — | — | 1 | 6.19 |
| CHEMBL1488229 | — | — | 1 | 6.16 |
| CHEMBL1388599 | — | — | 1 | 6.16 |
| CHEMBL1469670 | — | — | 1 | 6.14 |
| CHEMBL1392403 | — | — | 1 | 6.14 |
| CHEMBL1452159 | — | — | 1 | 6.12 |
| CHEMBL1463050 | — | — | 1 | 6.12 |
| CHEMBL1472681 | — | — | 1 | 6.11 |
| CHEMBL1416637 | — | — | 1 | 6.09 |
| CHEMBL1497295 | — | — | 1 | 6.07 |
| CHEMBL3211093 | — | — | 1 | 6.06 |
| CHEMBL1409822 | — | — | 1 | 6.05 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1350077 | — | IC50 | = | 180.0 | nM | 6.75 |
| CHEMBL1965654 | — | IC50 | = | 208.0 | nM | 6.68 |
| CHEMBL1300766 | — | IC50 | = | 220.0 | nM | 6.66 |
| CHEMBL1559811 | — | IC50 | = | 230.0 | nM | 6.64 |
| CHEMBL1528660 | — | IC50 | = | 240.0 | nM | 6.62 |
| CHEMBL1305304 | — | IC50 | = | 250.0 | nM | 6.60 |
| CHEMBL1320514 | — | IC50 | = | 260.0 | nM | 6.58 |
| CHEMBL1352270 | — | IC50 | = | 330.0 | nM | 6.48 |
| CHEMBL1505655 | — | IC50 | = | 330.0 | nM | 6.48 |
| CHEMBL1484661 | — | IC50 | = | 340.0 | nM | 6.47 |
| CHEMBL1418371 | — | IC50 | = | 360.0 | nM | 6.44 |
| CHEMBL1521793 | — | IC50 | = | 390.0 | nM | 6.41 |
| CHEMBL1302818 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL1369231 | — | IC50 | = | 460.0 | nM | 6.34 |
| CHEMBL1351755 | — | IC50 | = | 470.0 | nM | 6.33 |
| CHEMBL1393156 | — | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL1465119 | — | IC50 | = | 580.0 | nM | 6.24 |
| CHEMBL1255937 | ANCITABINE HYDROCHLORIDE | IC50 | = | 640.0 | nM | 6.19 |
| CHEMBL1430068 | — | IC50 | = | 650.0 | nM | 6.19 |
| CHEMBL1388599 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL1488229 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL1392403 | — | IC50 | = | 720.0 | nM | 6.14 |
| CHEMBL1469670 | — | IC50 | = | 730.0 | nM | 6.14 |
| CHEMBL1452159 | — | IC50 | = | 760.0 | nM | 6.12 |
| CHEMBL1463050 | — | IC50 | = | 760.0 | nM | 6.12 |
| CHEMBL1472681 | — | IC50 | = | 780.0 | nM | 6.11 |
| CHEMBL1416637 | — | IC50 | = | 820.0 | nM | 6.09 |
| CHEMBL1497295 | — | IC50 | = | 850.0 | nM | 6.07 |
| CHEMBL3211093 | — | IC50 | = | 880.0 | nM | 6.06 |
| CHEMBL1409822 | — | IC50 | = | 890.0 | nM | 6.05 |
| CHEMBL1339546 | — | IC50 | = | 1020.0 | nM | 5.99 |
| CHEMBL1416848 | — | IC50 | = | 1070.0 | nM | 5.97 |
| CHEMBL1300952 | — | IC50 | = | 1060.0 | nM | 5.97 |
| CHEMBL1436389 | — | IC50 | = | 1130.0 | nM | 5.95 |
| CHEMBL1299637 | — | IC50 | = | 1130.0 | nM | 5.95 |
| CHEMBL3189237 | — | IC50 | = | 1180.0 | nM | 5.93 |
| CHEMBL1529687 | — | IC50 | = | 1170.0 | nM | 5.93 |
| CHEMBL1362588 | — | IC50 | = | 1190.0 | nM | 5.92 |
| CHEMBL1587181 | — | IC50 | = | 1270.0 | nM | 5.90 |
| CHEMBL1321622 | — | IC50 | = | 1260.0 | nM | 5.90 |
| CHEMBL1520650 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL1480464 | — | IC50 | = | 1280.0 | nM | 5.89 |
| CHEMBL1575588 | — | IC50 | = | 1310.0 | nM | 5.88 |
| CHEMBL1490048 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL1577938 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL1611371 | — | IC50 | = | 1420.0 | nM | 5.85 |
| CHEMBL1313238 | — | IC50 | = | 1460.0 | nM | 5.84 |
| CHEMBL1519454 | — | IC50 | = | 1480.0 | nM | 5.83 |
| CHEMBL1446437 | — | IC50 | = | 1480.0 | nM | 5.83 |
| CHEMBL1366006 | — | IC50 | = | 1520.0 | nM | 5.82 |