Assay Detail
Functional
CHEMBL1738171
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of UBC13 Polyubiquitin Inhibitors using a Bfl-1 counterscreen. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID485273, AID485343]
353
Total Activities
352
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 353 | 5.15 | 6.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1384172 | — | — | 1 | 6.44 |
| CHEMBL1310325 | — | — | 1 | 6.26 |
| CHEMBL1528814 | — | — | 1 | 5.96 |
| CHEMBL1343853 | — | — | 1 | 5.76 |
| CHEMBL1532679 | — | — | 1 | 5.70 |
| CHEMBL1984581 | — | — | 1 | 5.63 |
| CHEMBL1540627 | — | — | 1 | 5.52 |
| CHEMBL1981290 | — | — | 1 | 5.51 |
| CHEMBL1981063 | — | — | 1 | 5.51 |
| CHEMBL1576266 | — | — | 1 | 5.48 |
| CHEMBL1427763 | — | — | 1 | 5.46 |
| CHEMBL1995152 | — | — | 1 | 5.42 |
| CHEMBL1564990 | — | — | 1 | 5.39 |
| CHEMBL1986183 | — | — | 1 | 5.34 |
| CHEMBL1534034 | — | — | 1 | 5.31 |
| CHEMBL1973159 | — | — | 1 | 5.29 |
| CHEMBL1494737 | — | — | 1 | 5.28 |
| CHEMBL1989158 | — | — | 1 | 5.26 |
| CHEMBL1520667 | — | — | 1 | 5.24 |
| CHEMBL1487183 | ALEXIDINE HYDROCHLORIDE | — | 1 | 5.22 |
| CHEMBL1320463 | — | — | 1 | 5.21 |
| CHEMBL157351 | — | — | 1 | 5.21 |
| CHEMBL1208858 | CALMIDAZOLIUM CHLORIDE | — | 1 | 5.21 |
| CHEMBL1200883 | THONZONIUM BROMIDE | 4.0 | 1 | 5.19 |
| CHEMBL1442656 | — | — | 1 | 5.18 |
| CHEMBL1436792 | — | — | 1 | 5.16 |
| CHEMBL1592706 | — | — | 1 | 5.13 |
| CHEMBL1402190 | — | — | 1 | 5.10 |
| CHEMBL1589425 | — | — | 1 | 5.09 |
| CHEMBL1548086 | — | — | 1 | 5.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1384172 | — | IC50 | = | 360.0 | nM | 6.44 |
| CHEMBL1310325 | — | IC50 | = | 550.0 | nM | 6.26 |
| CHEMBL1528814 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL1343853 | — | IC50 | = | 1720.0 | nM | 5.76 |
| CHEMBL1532679 | — | IC50 | = | 2020.0 | nM | 5.70 |
| CHEMBL1984581 | — | IC50 | = | 2330.0 | nM | 5.63 |
| CHEMBL1540627 | — | IC50 | = | 2990.0 | nM | 5.52 |
| CHEMBL1981290 | — | IC50 | = | 3080.0 | nM | 5.51 |
| CHEMBL1981063 | — | IC50 | = | 3110.0 | nM | 5.51 |
| CHEMBL1576266 | — | IC50 | = | 3320.0 | nM | 5.48 |
| CHEMBL1427763 | — | IC50 | = | 3440.0 | nM | 5.46 |
| CHEMBL1995152 | — | IC50 | = | 3850.0 | nM | 5.42 |
| CHEMBL1564990 | — | IC50 | = | 4030.0 | nM | 5.39 |
| CHEMBL1986183 | — | IC50 | = | 4600.0 | nM | 5.34 |
| CHEMBL1534034 | — | IC50 | = | 4880.0 | nM | 5.31 |
| CHEMBL1973159 | — | IC50 | = | 5140.0 | nM | 5.29 |
| CHEMBL1494737 | — | IC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL1989158 | — | IC50 | = | 5510.0 | nM | 5.26 |
| CHEMBL1520667 | — | IC50 | = | 5820.0 | nM | 5.24 |
| CHEMBL1487183 | ALEXIDINE HYDROCHLORIDE | IC50 | = | 5950.0 | nM | 5.22 |
| CHEMBL157351 | — | IC50 | = | 6110.0 | nM | 5.21 |
| CHEMBL1320463 | — | IC50 | = | 6100.0 | nM | 5.21 |
| CHEMBL1208858 | CALMIDAZOLIUM CHLORIDE | IC50 | = | 6230.0 | nM | 5.21 |
| CHEMBL1200883 | THONZONIUM BROMIDE | IC50 | = | 6440.0 | nM | 5.19 |
| CHEMBL1442656 | — | IC50 | = | 6580.0 | nM | 5.18 |
| CHEMBL1436792 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL1592706 | — | IC50 | = | 7490.0 | nM | 5.13 |
| CHEMBL1402190 | — | IC50 | = | 8020.0 | nM | 5.10 |
| CHEMBL1589425 | — | IC50 | = | 8080.0 | nM | 5.09 |
| CHEMBL1548086 | — | IC50 | = | 8260.0 | nM | 5.08 |
| CHEMBL1456173 | — | IC50 | = | 8520.0 | nM | 5.07 |
| CHEMBL1316978 | — | IC50 | = | 8510.0 | nM | 5.07 |
| CHEMBL1509041 | — | IC50 | = | 8760.0 | nM | 5.06 |
| CHEMBL1448793 | — | IC50 | = | 9710.0 | nM | 5.01 |
| CHEMBL1317622 | — | IC50 | = | 9730.0 | nM | 5.01 |
| CHEMBL1316468 | — | IC50 | = | 10100.0 | nM | 5.00 |
| CHEMBL1509380 | — | IC50 | = | 10100.0 | nM | 5.00 |
| CHEMBL1226 | AMINODIMETHOXYQUINAZOLINYLPIPERAZINE | IC50 | = | 11100.0 | nM | 4.96 |
| CHEMBL1978733 | — | IC50 | = | 11400.0 | nM | 4.94 |
| CHEMBL1328456 | — | IC50 | = | 11700.0 | nM | 4.93 |
| CHEMBL1437186 | — | IC50 | = | 11800.0 | nM | 4.93 |
| CHEMBL1547025 | — | IC50 | = | 12400.0 | nM | 4.91 |
| CHEMBL1374245 | — | IC50 | = | 12500.0 | nM | 4.90 |
| CHEMBL591404 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL461579 | — | IC50 | = | 13200.0 | nM | 4.88 |
| CHEMBL1557893 | — | IC50 | = | 13300.0 | nM | 4.88 |
| CHEMBL1510761 | — | IC50 | = | 13100.0 | nM | 4.88 |
| CHEMBL1552992 | — | IC50 | = | 13900.0 | nM | 4.86 |
| CHEMBL1699641 | — | IC50 | = | 14200.0 | nM | 4.85 |
| CHEMBL1321398 | — | IC50 | = | 14900.0 | nM | 4.83 |