Assay Detail
Functional
CHEMBL1738183
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response confirmation of uHTS of chemical inhibitors of B-cell specific antigen receptor-induced NF-kB activation in a 697B cell line using a luminescence assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID435022, AID435025, AID465]
470
Total Activities
469
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 470 | 5.09 | 6.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1607086 | — | — | 1 | 6.80 |
| CHEMBL1453181 | — | — | 1 | 6.80 |
| CHEMBL1598445 | — | — | 1 | 6.80 |
| CHEMBL1559811 | — | — | 1 | 6.68 |
| CHEMBL1608382 | — | — | 1 | 6.60 |
| CHEMBL1497295 | — | — | 1 | 6.57 |
| CHEMBL1427350 | — | — | 1 | 6.57 |
| CHEMBL1312928 | — | — | 1 | 6.57 |
| CHEMBL1438842 | — | — | 1 | 6.55 |
| CHEMBL1431151 | — | — | 1 | 6.52 |
| CHEMBL1578584 | — | — | 1 | 6.50 |
| CHEMBL1452159 | — | — | 1 | 6.43 |
| CHEMBL1528660 | — | — | 1 | 6.41 |
| CHEMBL1445134 | — | — | 1 | 6.39 |
| CHEMBL1416637 | — | — | 1 | 6.38 |
| CHEMBL1393156 | — | — | 1 | 6.37 |
| CHEMBL1358180 | — | — | 1 | 6.36 |
| CHEMBL1472681 | — | — | 1 | 6.36 |
| CHEMBL1387790 | — | — | 1 | 6.26 |
| CHEMBL1430068 | — | — | 1 | 6.24 |
| CHEMBL1595476 | — | — | 1 | 6.23 |
| CHEMBL3189237 | — | — | 1 | 6.23 |
| CHEMBL1534546 | — | — | 1 | 6.20 |
| CHEMBL1573524 | — | — | 1 | 6.19 |
| CHEMBL1436389 | — | — | 1 | 6.17 |
| CHEMBL1465119 | — | — | 1 | 6.17 |
| CHEMBL1587181 | — | — | 1 | 6.17 |
| CHEMBL1469676 | — | — | 1 | 6.14 |
| CHEMBL1965654 | — | — | 1 | 6.13 |
| CHEMBL1422720 | — | — | 1 | 6.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1607086 | — | IC50 | = | 160.0 | nM | 6.80 |
| CHEMBL1453181 | — | IC50 | = | 160.0 | nM | 6.80 |
| CHEMBL1598445 | — | IC50 | = | 160.0 | nM | 6.80 |
| CHEMBL1559811 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL1608382 | — | IC50 | = | 250.0 | nM | 6.60 |
| CHEMBL1427350 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL1497295 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL1312928 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL1438842 | — | IC50 | = | 280.0 | nM | 6.55 |
| CHEMBL1431151 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL1578584 | — | IC50 | = | 320.0 | nM | 6.50 |
| CHEMBL1452159 | — | IC50 | = | 370.0 | nM | 6.43 |
| CHEMBL1528660 | — | IC50 | = | 390.0 | nM | 6.41 |
| CHEMBL1445134 | — | IC50 | = | 410.0 | nM | 6.39 |
| CHEMBL1416637 | — | IC50 | = | 420.0 | nM | 6.38 |
| CHEMBL1393156 | — | IC50 | = | 430.0 | nM | 6.37 |
| CHEMBL1472681 | — | IC50 | = | 440.0 | nM | 6.36 |
| CHEMBL1358180 | — | IC50 | = | 440.0 | nM | 6.36 |
| CHEMBL1387790 | — | IC50 | = | 550.0 | nM | 6.26 |
| CHEMBL1430068 | — | IC50 | = | 570.0 | nM | 6.24 |
| CHEMBL1595476 | — | IC50 | = | 590.0 | nM | 6.23 |
| CHEMBL3189237 | — | IC50 | = | 590.0 | nM | 6.23 |
| CHEMBL1534546 | — | IC50 | = | 630.0 | nM | 6.20 |
| CHEMBL1573524 | — | IC50 | = | 640.0 | nM | 6.19 |
| CHEMBL1587181 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL1436389 | — | IC50 | = | 670.0 | nM | 6.17 |
| CHEMBL1465119 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL1469676 | — | IC50 | = | 720.0 | nM | 6.14 |
| CHEMBL1965654 | — | IC50 | = | 740.0 | nM | 6.13 |
| CHEMBL1422720 | — | IC50 | = | 790.0 | nM | 6.10 |
| CHEMBL1575588 | — | IC50 | = | 790.0 | nM | 6.10 |
| CHEMBL1521793 | — | IC50 | = | 820.0 | nM | 6.09 |
| CHEMBL1428662 | — | IC50 | = | 850.0 | nM | 6.07 |
| CHEMBL1351755 | — | IC50 | = | 850.0 | nM | 6.07 |
| CHEMBL1350077 | — | IC50 | = | 930.0 | nM | 6.03 |
| CHEMBL1321622 | — | IC50 | = | 1130.0 | nM | 5.95 |
| CHEMBL1352850 | — | IC50 | = | 1120.0 | nM | 5.95 |
| CHEMBL1469670 | — | IC50 | = | 1130.0 | nM | 5.95 |
| CHEMBL1403324 | — | IC50 | = | 1240.0 | nM | 5.91 |
| CHEMBL1369231 | — | IC50 | = | 1230.0 | nM | 5.91 |
| CHEMBL1890899 | — | IC50 | = | 1220.0 | nM | 5.91 |
| CHEMBL1409822 | — | IC50 | = | 1260.0 | nM | 5.90 |
| CHEMBL3189935 | — | IC50 | = | 1250.0 | nM | 5.90 |
| CHEMBL1339546 | — | IC50 | = | 1250.0 | nM | 5.90 |
| CHEMBL1409900 | — | IC50 | = | 1270.0 | nM | 5.90 |
| CHEMBL1328161 | — | IC50 | = | 1290.0 | nM | 5.89 |
| CHEMBL1378086 | — | IC50 | = | 1330.0 | nM | 5.88 |
| CHEMBL1611371 | — | IC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL1302375 | — | IC50 | = | 1350.0 | nM | 5.87 |
| CHEMBL1301144 | — | IC50 | = | 1360.0 | nM | 5.87 |