Assay Detail
Functional
CHEMBL1738425
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR Analysis of Antagonists of the MOR Receptor using an Image-Based Assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1777, AID1785, AID1786, AID1966, AID2133, AID2136, AID2284, AID2285, AID2478, AID488842]
62
Total Activities
62
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 62 | 5.61 | 6.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1369123 | — | — | 1 | 6.05 |
| CHEMBL1511139 | — | — | 1 | 5.72 |
| CHEMBL1461661 | — | — | 1 | 5.07 |
| CHEMBL1455766 | — | — | 1 | - |
| CHEMBL1716867 | — | — | 1 | - |
| CHEMBL1707460 | — | — | 1 | - |
| CHEMBL1416769 | — | — | 1 | - |
| CHEMBL1490629 | — | — | 1 | - |
| CHEMBL1726168 | — | — | 1 | - |
| CHEMBL1706477 | — | — | 1 | - |
| CHEMBL1405968 | — | — | 1 | - |
| CHEMBL1565651 | — | — | 1 | - |
| CHEMBL1359415 | — | — | 1 | - |
| CHEMBL1705910 | — | — | 1 | - |
| CHEMBL1724710 | — | — | 1 | - |
| CHEMBL1342964 | — | — | 1 | - |
| CHEMBL1731800 | — | — | 1 | - |
| CHEMBL1371990 | — | — | 1 | - |
| CHEMBL1732148 | — | — | 1 | - |
| CHEMBL1712643 | — | — | 1 | - |
| CHEMBL1480657 | — | — | 1 | - |
| CHEMBL1455762 | — | — | 1 | - |
| CHEMBL1348399 | — | — | 1 | - |
| CHEMBL1346675 | — | — | 1 | - |
| CHEMBL1508445 | — | — | 1 | - |
| CHEMBL1726942 | — | — | 1 | - |
| CHEMBL1440728 | — | — | 1 | - |
| CHEMBL1723909 | — | — | 1 | - |
| CHEMBL1594497 | — | — | 1 | - |
| CHEMBL1493095 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1369123 | — | IC50 | = | 897.0 | nM | 6.05 |
| CHEMBL1511139 | — | IC50 | = | 1920.0 | nM | 5.72 |
| CHEMBL1461661 | — | IC50 | = | 8430.0 | nM | 5.07 |
| CHEMBL1707460 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1710618 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1716867 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1455766 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1362498 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1455045 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1430337 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1568059 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1430524 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1718305 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1343080 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1417841 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1569631 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1719035 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1384726 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1493386 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1585267 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1564473 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1588996 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1478375 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1729385 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1403666 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1720217 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1732148 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1493095 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1594497 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1723909 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1440728 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1726942 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1508445 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1346675 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1348399 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1455762 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1480657 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1712643 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1416769 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1371990 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1731800 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1342964 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1724710 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1705910 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1359415 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1565651 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1405968 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1706477 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1726168 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1490629 | — | IC50 | > | 32000.0 | nM | - |