Assay Detail
Functional
CHEMBL1738438
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of uHTS small molecule inhibitors of tim10-1: a luminescent TIM10 yeast counterscreen. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID463190, AID463194, AID493003]
145
Total Activities
145
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Saccharomyces cerevisiae S288c |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Mitochondrial import inner membrane translocase subunit TIM10 (CHEMBL1741194) ↗| Type | SINGLE PROTEIN |
| Organism | Saccharomyces cerevisiae S288c |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 145 | 5.33 | 6.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1421736 | — | — | 1 | 6.58 |
| CHEMBL3199050 | — | — | 1 | 6.58 |
| CHEMBL1519298 | — | — | 1 | 6.39 |
| CHEMBL51085 | EBSELEN | 3.0 | 1 | 6.24 |
| CHEMBL1515506 | — | — | 1 | 6.18 |
| CHEMBL1485605 | — | — | 1 | 6.16 |
| CHEMBL1505636 | — | — | 1 | 6.13 |
| CHEMBL1353110 | — | — | 1 | 6.10 |
| CHEMBL1376392 | — | — | 1 | 6.06 |
| CHEMBL1485010 | — | — | 1 | 5.94 |
| CHEMBL1549175 | — | — | 1 | 5.92 |
| CHEMBL1995800 | — | — | 1 | 5.91 |
| CHEMBL1470485 | — | — | 1 | 5.90 |
| CHEMBL1391098 | — | — | 1 | 5.89 |
| CHEMBL211969 | — | — | 1 | 5.88 |
| CHEMBL1561609 | — | — | 1 | 5.86 |
| CHEMBL1303810 | — | — | 1 | 5.85 |
| CHEMBL1407254 | — | — | 1 | 5.83 |
| CHEMBL1450616 | — | — | 1 | 5.76 |
| CHEMBL1471900 | — | — | 1 | 5.76 |
| CHEMBL1371138 | — | — | 1 | 5.74 |
| CHEMBL1984894 | — | — | 1 | 5.73 |
| CHEMBL1518799 | — | — | 1 | 5.72 |
| CHEMBL1549738 | — | — | 1 | 5.70 |
| CHEMBL3213220 | — | — | 1 | 5.64 |
| CHEMBL1463422 | — | — | 1 | 5.64 |
| CHEMBL1467732 | — | — | 1 | 5.64 |
| CHEMBL1401698 | — | — | 1 | 5.63 |
| CHEMBL1495590 | — | — | 1 | 5.62 |
| CHEMBL1459930 | — | — | 1 | 5.62 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1421736 | — | IC50 | = | 260.0 | nM | 6.58 |
| CHEMBL3199050 | — | IC50 | = | 260.0 | nM | 6.58 |
| CHEMBL1519298 | — | IC50 | = | 410.0 | nM | 6.39 |
| CHEMBL51085 | EBSELEN | IC50 | = | 580.0 | nM | 6.24 |
| CHEMBL1515506 | — | IC50 | = | 660.0 | nM | 6.18 |
| CHEMBL1485605 | — | IC50 | = | 690.0 | nM | 6.16 |
| CHEMBL1505636 | — | IC50 | = | 740.0 | nM | 6.13 |
| CHEMBL1353110 | — | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL1376392 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL1485010 | — | IC50 | = | 1150.0 | nM | 5.94 |
| CHEMBL1549175 | — | IC50 | = | 1190.0 | nM | 5.92 |
| CHEMBL1995800 | — | IC50 | = | 1220.0 | nM | 5.91 |
| CHEMBL1470485 | — | IC50 | = | 1270.0 | nM | 5.90 |
| CHEMBL1391098 | — | IC50 | = | 1280.0 | nM | 5.89 |
| CHEMBL211969 | — | IC50 | = | 1330.0 | nM | 5.88 |
| CHEMBL1561609 | — | IC50 | = | 1390.0 | nM | 5.86 |
| CHEMBL1303810 | — | IC50 | = | 1410.0 | nM | 5.85 |
| CHEMBL1407254 | — | IC50 | = | 1490.0 | nM | 5.83 |
| CHEMBL1471900 | — | IC50 | = | 1740.0 | nM | 5.76 |
| CHEMBL1450616 | — | IC50 | = | 1720.0 | nM | 5.76 |
| CHEMBL1371138 | — | IC50 | = | 1820.0 | nM | 5.74 |
| CHEMBL1984894 | — | IC50 | = | 1870.0 | nM | 5.73 |
| CHEMBL1518799 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL1549738 | — | IC50 | = | 1980.0 | nM | 5.70 |
| CHEMBL3213220 | — | IC50 | = | 2280.0 | nM | 5.64 |
| CHEMBL1467732 | — | IC50 | = | 2270.0 | nM | 5.64 |
| CHEMBL1463422 | — | IC50 | = | 2280.0 | nM | 5.64 |
| CHEMBL1401698 | — | IC50 | = | 2350.0 | nM | 5.63 |
| CHEMBL1459930 | — | IC50 | = | 2390.0 | nM | 5.62 |
| CHEMBL1495590 | — | IC50 | = | 2420.0 | nM | 5.62 |
| CHEMBL1562493 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL1447783 | — | IC50 | = | 2610.0 | nM | 5.58 |
| CHEMBL1574219 | — | IC50 | = | 2720.0 | nM | 5.57 |
| CHEMBL1363382 | — | IC50 | = | 2890.0 | nM | 5.54 |
| CHEMBL1384790 | — | IC50 | = | 2910.0 | nM | 5.54 |
| CHEMBL3198175 | — | IC50 | = | 2940.0 | nM | 5.53 |
| CHEMBL1335988 | — | IC50 | = | 2990.0 | nM | 5.52 |
| CHEMBL1503238 | — | IC50 | = | 3090.0 | nM | 5.51 |
| CHEMBL1718013 | — | IC50 | = | 3150.0 | nM | 5.50 |
| CHEMBL1368514 | — | IC50 | = | 3190.0 | nM | 5.50 |
| CHEMBL1554169 | — | IC50 | = | 3320.0 | nM | 5.48 |
| CHEMBL1372447 | — | IC50 | = | 3320.0 | nM | 5.48 |
| CHEMBL1610316 | — | IC50 | = | 3490.0 | nM | 5.46 |
| CHEMBL1304513 | — | IC50 | = | 3430.0 | nM | 5.46 |
| CHEMBL1324805 | — | IC50 | = | 3620.0 | nM | 5.44 |
| CHEMBL1988138 | — | IC50 | = | 3660.0 | nM | 5.44 |
| CHEMBL1964878 | — | IC50 | = | 3810.0 | nM | 5.42 |
| CHEMBL3192555 | — | IC50 | = | 3940.0 | nM | 5.41 |
| CHEMBL1572280 | — | IC50 | = | 3920.0 | nM | 5.41 |
| CHEMBL1544036 | — | IC50 | = | 3860.0 | nM | 5.41 |