Assay Detail
Functional
CHEMBL1738447
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response of TOR pathway GFP-fusion proteins in Saccharomyces cerevisiae specifically MEP2 based on MLPCN hits. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1908, AID488812, AID488818]
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Saccharomyces cerevisiae |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Ammonium transporter MEP2 (CHEMBL1741183) ↗| Type | SINGLE PROTEIN |
| Organism | Saccharomyces cerevisiae S288c |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 12 | 5.52 | 5.98 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1458319 | — | — | 1 | 5.98 |
| CHEMBL1562104 | — | — | 1 | 5.91 |
| CHEMBL518292 | ISOVELLERAL | — | 1 | 5.90 |
| CHEMBL1590745 | — | — | 1 | 5.86 |
| CHEMBL1430795 | — | — | 1 | 5.64 |
| CHEMBL1344927 | — | — | 1 | 5.52 |
| CHEMBL1581772 | — | — | 1 | 5.41 |
| CHEMBL1505372 | — | — | 1 | 5.17 |
| CHEMBL1578341 | — | — | 1 | 4.90 |
| CHEMBL1336054 | — | — | 1 | 4.86 |
| CHEMBL1318350 | — | — | 1 | - |
| CHEMBL1990694 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1458319 | — | EC50 | = | 1042.0 | nM | 5.98 |
| CHEMBL1562104 | — | EC50 | = | 1226.0 | nM | 5.91 |
| CHEMBL518292 | ISOVELLERAL | EC50 | = | 1264.0 | nM | 5.90 |
| CHEMBL1590745 | — | EC50 | = | 1381.0 | nM | 5.86 |
| CHEMBL1430795 | — | EC50 | = | 2277.0 | nM | 5.64 |
| CHEMBL1344927 | — | EC50 | = | 3006.0 | nM | 5.52 |
| CHEMBL1581772 | — | EC50 | = | 3857.0 | nM | 5.41 |
| CHEMBL1505372 | — | EC50 | = | 6846.0 | nM | 5.17 |
| CHEMBL1578341 | — | EC50 | = | 12710.0 | nM | 4.90 |
| CHEMBL1336054 | — | EC50 | = | 13690.0 | nM | 4.86 |
| CHEMBL1318350 | — | EC50 | > | 33000.0 | nM | - |
| CHEMBL1990694 | — | EC50 | > | 33000.0 | nM | - |