Assay Detail
Binding
CHEMBL1738581
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR LYP1 Fluorescent Assay using OMFP substrate for In Vitro dose response studies. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1779, AID1784, AID2686, AID449726, AID488869]
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Tyrosine-protein phosphatase non-receptor type 22 (CHEMBL2889) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 4.74 | 5.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1701224 | — | — | 1 | 5.22 |
| CHEMBL1438889 | — | — | 1 | 5.13 |
| CHEMBL1443268 | — | — | 1 | 5.11 |
| CHEMBL1710150 | — | — | 1 | 4.96 |
| CHEMBL1492305 | — | — | 1 | 4.79 |
| CHEMBL1371816 | — | — | 1 | 4.47 |
| CHEMBL1698734 | — | — | 1 | 4.36 |
| CHEMBL1417070 | — | — | 1 | 4.32 |
| CHEMBL1439815 | — | — | 1 | 4.29 |
| CHEMBL1718018 | — | — | 1 | - |
| CHEMBL1700415 | — | — | 1 | - |
| CHEMBL1721448 | — | — | 1 | - |
| CHEMBL1713374 | — | — | 1 | - |
| CHEMBL1714966 | — | — | 1 | - |
| CHEMBL1706168 | — | — | 1 | - |
| CHEMBL1735637 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1701224 | — | IC50 | = | 6069.0 | nM | 5.22 |
| CHEMBL1438889 | — | IC50 | = | 7461.0 | nM | 5.13 |
| CHEMBL1443268 | — | IC50 | = | 7713.0 | nM | 5.11 |
| CHEMBL1710150 | — | IC50 | = | 10955.0 | nM | 4.96 |
| CHEMBL1492305 | — | IC50 | = | 16047.0 | nM | 4.79 |
| CHEMBL1371816 | — | IC50 | = | 34166.0 | nM | 4.47 |
| CHEMBL1698734 | — | IC50 | = | 43409.0 | nM | 4.36 |
| CHEMBL1417070 | — | IC50 | = | 47399.0 | nM | 4.32 |
| CHEMBL1439815 | — | IC50 | = | 50909.0 | nM | 4.29 |
| CHEMBL1718018 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1700415 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1721448 | — | IC50 | = | 139495.0 | nM | - |
| CHEMBL1713374 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL1714966 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1706168 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1735637 | — | IC50 | > | 100000.0 | nM | - |