Assay Detail
Functional
CHEMBL1738596
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR LYP1 Fluorescent Assay using OMFP substrate for In Vitro dose response studies - Set 2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1779, AID1784, AID2140, AID449726, AID488869]
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Tyrosine-protein phosphatase non-receptor type 22 (CHEMBL2889) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 34 | 5.08 | 5.97 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1438889 | — | — | 1 | 5.97 |
| CHEMBL1701224 | — | — | 1 | 5.91 |
| CHEMBL1320181 | — | — | 1 | 5.81 |
| CHEMBL1390354 | — | — | 1 | 5.71 |
| CHEMBL1443268 | — | — | 1 | 5.50 |
| CHEMBL1371816 | — | — | 1 | 5.42 |
| CHEMBL1492305 | — | — | 1 | 5.41 |
| CHEMBL1704862 | — | — | 1 | 5.39 |
| CHEMBL1439815 | — | — | 1 | 5.34 |
| CHEMBL1550429 | — | — | 1 | 5.32 |
| CHEMBL1456664 | — | — | 1 | 5.29 |
| CHEMBL1572439 | — | — | 1 | 5.28 |
| CHEMBL1719149 | — | — | 1 | 5.25 |
| CHEMBL1724482 | — | — | 1 | 4.86 |
| CHEMBL1722719 | — | — | 1 | 4.84 |
| CHEMBL1562411 | — | — | 1 | 4.83 |
| CHEMBL1718018 | — | — | 1 | 4.66 |
| CHEMBL1706168 | — | — | 1 | 4.45 |
| CHEMBL1417070 | — | — | 1 | 4.36 |
| CHEMBL1714966 | — | — | 1 | 4.18 |
| CHEMBL1732934 | — | — | 1 | 4.02 |
| CHEMBL1700415 | — | — | 1 | 4.00 |
| CHEMBL1719458 | — | — | 1 | - |
| CHEMBL1478943 | — | — | 1 | - |
| CHEMBL1461397 | — | — | 1 | - |
| CHEMBL1735637 | — | — | 1 | - |
| CHEMBL1488869 | — | — | 1 | - |
| CHEMBL1425801 | — | — | 1 | - |
| CHEMBL1715912 | — | — | 1 | - |
| CHEMBL1729772 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1438889 | — | IC50 | = | 1080.0 | nM | 5.97 |
| CHEMBL1701224 | — | IC50 | = | 1240.0 | nM | 5.91 |
| CHEMBL1320181 | — | IC50 | = | 1540.0 | nM | 5.81 |
| CHEMBL1390354 | — | IC50 | = | 1940.0 | nM | 5.71 |
| CHEMBL1443268 | — | IC50 | = | 3150.0 | nM | 5.50 |
| CHEMBL1371816 | — | IC50 | = | 3770.0 | nM | 5.42 |
| CHEMBL1492305 | — | IC50 | = | 3920.0 | nM | 5.41 |
| CHEMBL1704862 | — | IC50 | = | 4040.0 | nM | 5.39 |
| CHEMBL1439815 | — | IC50 | = | 4560.0 | nM | 5.34 |
| CHEMBL1550429 | — | IC50 | = | 4780.0 | nM | 5.32 |
| CHEMBL1456664 | — | IC50 | = | 5130.0 | nM | 5.29 |
| CHEMBL1572439 | — | IC50 | = | 5270.0 | nM | 5.28 |
| CHEMBL1719149 | — | IC50 | = | 5670.0 | nM | 5.25 |
| CHEMBL1724482 | — | IC50 | = | 13700.0 | nM | 4.86 |
| CHEMBL1722719 | — | IC50 | = | 14600.0 | nM | 4.84 |
| CHEMBL1562411 | — | IC50 | = | 14700.0 | nM | 4.83 |
| CHEMBL1718018 | — | IC50 | = | 21800.0 | nM | 4.66 |
| CHEMBL1706168 | — | IC50 | = | 35500.0 | nM | 4.45 |
| CHEMBL1417070 | — | IC50 | = | 43700.0 | nM | 4.36 |
| CHEMBL1714966 | — | IC50 | = | 65500.0 | nM | 4.18 |
| CHEMBL1732934 | — | IC50 | = | 95300.0 | nM | 4.02 |
| CHEMBL1700415 | — | IC50 | = | 99100.0 | nM | 4.00 |
| CHEMBL1719458 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1478943 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1461397 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1735637 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1488869 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1425801 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1715912 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1729772 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1710376 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1400747 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1721448 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1713374 | — | IC50 | > | 100000.0 | nM | - |