Assay Detail
Functional
CHEMBL1738609
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR VHR1 Fluorescent Assay for In Vitro dose response studies Set 2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1654, AID1661, AID1878]
84
Total Activities
83
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Dual specificity protein phosphatase 3 (CHEMBL2635) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 84 | 5.01 | 7.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1460470 | — | — | 2 | 7.08 |
| CHEMBL1322542 | — | — | 1 | 6.84 |
| CHEMBL1385949 | — | — | 1 | 6.67 |
| CHEMBL1445488 | — | — | 1 | 6.66 |
| CHEMBL1393151 | — | — | 1 | 6.65 |
| CHEMBL1304193 | — | — | 1 | 6.58 |
| CHEMBL1408579 | — | — | 1 | 6.46 |
| CHEMBL1605172 | — | — | 1 | 6.40 |
| CHEMBL1732016 | — | — | 1 | 6.32 |
| CHEMBL1505246 | — | — | 1 | 6.02 |
| CHEMBL1447397 | — | — | 1 | 5.77 |
| CHEMBL601167 | — | — | 1 | 5.60 |
| CHEMBL1373210 | — | — | 1 | 5.45 |
| CHEMBL1730304 | — | — | 1 | 5.32 |
| CHEMBL1569076 | — | — | 1 | 5.27 |
| CHEMBL1304974 | — | — | 1 | 4.91 |
| CHEMBL1711927 | — | — | 1 | 4.87 |
| CHEMBL1369492 | — | — | 1 | 4.82 |
| CHEMBL1704720 | — | — | 1 | 4.82 |
| CHEMBL1597485 | — | — | 1 | 4.81 |
| CHEMBL1708762 | — | — | 1 | 4.79 |
| CHEMBL1721618 | — | — | 1 | 4.75 |
| CHEMBL1343331 | — | — | 1 | 4.72 |
| CHEMBL1730959 | — | — | 1 | 4.71 |
| CHEMBL1704444 | — | — | 1 | 4.52 |
| CHEMBL1709810 | — | — | 1 | 4.50 |
| CHEMBL1710168 | — | — | 1 | 4.48 |
| CHEMBL1724311 | — | — | 1 | 4.47 |
| CHEMBL1723290 | — | — | 1 | 4.42 |
| CHEMBL1699305 | — | — | 1 | 4.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1460470 | — | IC50 | = | 82.8 | nM | 7.08 |
| CHEMBL1322542 | — | IC50 | = | 143.0 | nM | 6.84 |
| CHEMBL1385949 | — | IC50 | = | 216.0 | nM | 6.67 |
| CHEMBL1445488 | — | IC50 | = | 218.0 | nM | 6.66 |
| CHEMBL1393151 | — | IC50 | = | 226.0 | nM | 6.65 |
| CHEMBL1304193 | — | IC50 | = | 260.0 | nM | 6.58 |
| CHEMBL1408579 | — | IC50 | = | 347.0 | nM | 6.46 |
| CHEMBL1605172 | — | IC50 | = | 402.0 | nM | 6.40 |
| CHEMBL1732016 | — | IC50 | = | 480.0 | nM | 6.32 |
| CHEMBL1505246 | — | IC50 | = | 960.0 | nM | 6.02 |
| CHEMBL1447397 | — | IC50 | = | 1690.0 | nM | 5.77 |
| CHEMBL601167 | — | IC50 | = | 2490.0 | nM | 5.60 |
| CHEMBL1373210 | — | IC50 | = | 3550.0 | nM | 5.45 |
| CHEMBL1730304 | — | IC50 | = | 4830.0 | nM | 5.32 |
| CHEMBL1569076 | — | IC50 | = | 5380.0 | nM | 5.27 |
| CHEMBL1304974 | — | IC50 | = | 12300.0 | nM | 4.91 |
| CHEMBL1711927 | — | IC50 | = | 13500.0 | nM | 4.87 |
| CHEMBL1369492 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL1704720 | — | IC50 | = | 15100.0 | nM | 4.82 |
| CHEMBL1597485 | — | IC50 | = | 15400.0 | nM | 4.81 |
| CHEMBL1708762 | — | IC50 | = | 16200.0 | nM | 4.79 |
| CHEMBL1721618 | — | IC50 | = | 17900.0 | nM | 4.75 |
| CHEMBL1343331 | — | IC50 | = | 18900.0 | nM | 4.72 |
| CHEMBL1730959 | — | IC50 | = | 19300.0 | nM | 4.71 |
| CHEMBL1704444 | — | IC50 | = | 30500.0 | nM | 4.52 |
| CHEMBL1709810 | — | IC50 | = | 31900.0 | nM | 4.50 |
| CHEMBL1710168 | — | IC50 | = | 32800.0 | nM | 4.48 |
| CHEMBL1724311 | — | IC50 | = | 33800.0 | nM | 4.47 |
| CHEMBL1723290 | — | IC50 | = | 38100.0 | nM | 4.42 |
| CHEMBL1699305 | — | IC50 | = | 40900.0 | nM | 4.39 |
| CHEMBL1724547 | — | IC50 | = | 41100.0 | nM | 4.39 |
| CHEMBL1735969 | — | IC50 | = | 47000.0 | nM | 4.33 |
| CHEMBL1733159 | — | IC50 | = | 48400.0 | nM | 4.32 |
| CHEMBL1702302 | — | IC50 | = | 60800.0 | nM | 4.22 |
| CHEMBL1421461 | — | IC50 | = | 61200.0 | nM | 4.21 |
| CHEMBL1720016 | — | IC50 | = | 65200.0 | nM | 4.19 |
| CHEMBL1733162 | — | IC50 | = | 67400.0 | nM | 4.17 |
| CHEMBL1723513 | — | IC50 | = | 67200.0 | nM | 4.17 |
| CHEMBL1714887 | — | IC50 | = | 71700.0 | nM | 4.14 |
| CHEMBL1455260 | — | IC50 | = | 76500.0 | nM | 4.12 |
| CHEMBL1519586 | — | IC50 | = | 78000.0 | nM | 4.11 |
| CHEMBL1301020 | — | IC50 | = | 85500.0 | nM | 4.07 |
| CHEMBL1716347 | — | IC50 | = | 86900.0 | nM | 4.06 |
| CHEMBL1461661 | — | IC50 | = | 90000.0 | nM | 4.05 |
| CHEMBL1719539 | — | IC50 | = | 99500.0 | nM | 4.00 |
| CHEMBL1736022 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1578067 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1425948 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1716867 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1735408 | — | IC50 | > | 100000.0 | nM | - |