Assay Detail
Functional
CHEMBL1738643
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for AddAB inhibitors: absorbance-based bacterial cell-based high throughput dose response assay for inhibitors of bacterial viability. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID435030, AID449728, AID449731, AID488942, AID488955, AID488956]
225
Total Activities
223
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 225 | 4.42 | 5.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL570105 | — | — | 1 | 5.48 |
| CHEMBL318153 | EDOXUDINE | 2.0 | 2 | 4.84 |
| CHEMBL1967099 | — | — | 1 | 4.83 |
| CHEMBL1502014 | — | — | 1 | 4.82 |
| CHEMBL3195943 | — | — | 1 | 4.78 |
| CHEMBL1546374 | — | — | 1 | 4.77 |
| CHEMBL1729758 | — | — | 1 | 4.76 |
| CHEMBL1396209 | — | — | 1 | 4.73 |
| CHEMBL1724246 | — | — | 1 | 4.68 |
| CHEMBL1428883 | — | — | 1 | 4.66 |
| CHEMBL1423626 | — | — | 1 | 4.66 |
| CHEMBL1414846 | — | — | 1 | 4.57 |
| CHEMBL443 | SULFAMETHOXAZOLE | 4.0 | 1 | 4.54 |
| CHEMBL1396843 | — | — | 1 | 4.54 |
| CHEMBL1584024 | — | — | 1 | 4.53 |
| CHEMBL1256400 | XYLOMETAZOLINE HYDROCHLORIDE | -1.0 | 1 | 4.53 |
| CHEMBL1447058 | — | — | 1 | 4.50 |
| CHEMBL3194778 | — | — | 1 | 4.50 |
| CHEMBL1989750 | — | — | 1 | 4.49 |
| CHEMBL415879 | PHENANTHROLINE | — | 1 | 4.45 |
| CHEMBL1588926 | — | — | 1 | 4.45 |
| CHEMBL1479316 | — | — | 1 | 4.45 |
| CHEMBL1528900 | — | — | 1 | 4.44 |
| CHEMBL1382917 | — | — | 1 | 4.43 |
| CHEMBL1431189 | — | — | 1 | 4.41 |
| CHEMBL1330558 | — | — | 1 | 4.38 |
| CHEMBL1476029 | — | — | 1 | 4.37 |
| CHEMBL3190283 | — | — | 1 | 4.34 |
| CHEMBL1407684 | — | — | 1 | 4.34 |
| CHEMBL1557648 | — | — | 1 | 4.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL570105 | — | IC50 | = | 3325.0 | nM | 5.48 |
| CHEMBL318153 | EDOXUDINE | IC50 | = | 14493.0 | nM | 4.84 |
| CHEMBL1967099 | — | IC50 | = | 14947.0 | nM | 4.83 |
| CHEMBL1502014 | — | IC50 | = | 15110.0 | nM | 4.82 |
| CHEMBL3195943 | — | IC50 | = | 16580.0 | nM | 4.78 |
| CHEMBL1546374 | — | IC50 | = | 16854.0 | nM | 4.77 |
| CHEMBL1729758 | — | IC50 | = | 17503.0 | nM | 4.76 |
| CHEMBL318153 | EDOXUDINE | IC50 | = | 18504.0 | nM | 4.73 |
| CHEMBL1396209 | — | IC50 | = | 18520.0 | nM | 4.73 |
| CHEMBL1724246 | — | IC50 | = | 21029.0 | nM | 4.68 |
| CHEMBL1428883 | — | IC50 | = | 22045.0 | nM | 4.66 |
| CHEMBL1423626 | — | IC50 | = | 21708.0 | nM | 4.66 |
| CHEMBL1414846 | — | IC50 | = | 27070.0 | nM | 4.57 |
| CHEMBL443 | SULFAMETHOXAZOLE | IC50 | = | 29167.0 | nM | 4.54 |
| CHEMBL1396843 | — | IC50 | = | 29010.0 | nM | 4.54 |
| CHEMBL1256400 | XYLOMETAZOLINE HYDROCHLORIDE | IC50 | = | 29687.0 | nM | 4.53 |
| CHEMBL1584024 | — | IC50 | = | 29870.0 | nM | 4.53 |
| CHEMBL1447058 | — | IC50 | = | 31941.0 | nM | 4.50 |
| CHEMBL3194778 | — | IC50 | = | 31838.0 | nM | 4.50 |
| CHEMBL1989750 | — | IC50 | = | 32235.0 | nM | 4.49 |
| CHEMBL415879 | PHENANTHROLINE | IC50 | = | 35186.0 | nM | 4.45 |
| CHEMBL1588926 | — | IC50 | = | 35780.0 | nM | 4.45 |
| CHEMBL1479316 | — | IC50 | = | 35604.0 | nM | 4.45 |
| CHEMBL1528900 | — | IC50 | = | 36544.0 | nM | 4.44 |
| CHEMBL1382917 | — | IC50 | = | 37456.0 | nM | 4.43 |
| CHEMBL1431189 | — | IC50 | = | 39007.0 | nM | 4.41 |
| CHEMBL1330558 | — | IC50 | = | 41484.0 | nM | 4.38 |
| CHEMBL1476029 | — | IC50 | = | 42780.0 | nM | 4.37 |
| CHEMBL1407684 | — | IC50 | = | 45862.0 | nM | 4.34 |
| CHEMBL3190283 | — | IC50 | = | 45933.0 | nM | 4.34 |
| CHEMBL1557648 | — | IC50 | = | 46958.0 | nM | 4.33 |
| CHEMBL2004847 | — | IC50 | = | 55530.0 | nM | 4.25 |
| CHEMBL1430038 | — | IC50 | = | 60237.0 | nM | 4.22 |
| CHEMBL1483355 | — | IC50 | = | 61670.0 | nM | 4.21 |
| CHEMBL1532238 | — | IC50 | = | 61057.0 | nM | 4.21 |
| CHEMBL1454721 | — | IC50 | = | 63768.0 | nM | 4.20 |
| CHEMBL1605292 | — | IC50 | = | 64886.0 | nM | 4.19 |
| CHEMBL1605805 | — | IC50 | = | 66128.0 | nM | 4.18 |
| CHEMBL1461482 | — | IC50 | = | 69657.0 | nM | 4.16 |
| CHEMBL1728955 | — | IC50 | = | 75900.0 | nM | 4.12 |
| CHEMBL67311 | — | IC50 | = | 77581.0 | nM | 4.11 |
| CHEMBL1559564 | — | IC50 | = | 83563.0 | nM | 4.08 |
| CHEMBL32793 | — | IC50 | = | 85187.0 | nM | 4.07 |
| CHEMBL1999960 | — | IC50 | = | 91436.0 | nM | 4.04 |
| CHEMBL1380414 | — | IC50 | = | 92632.0 | nM | 4.03 |
| CHEMBL1585527 | — | IC50 | = | 95304.0 | nM | 4.02 |
| CHEMBL1342357 | — | IC50 | = | 96776.0 | nM | 4.01 |
| CHEMBL1998606 | — | IC50 | = | 98169.0 | nM | 4.01 |
| CHEMBL81782 | — | IC50 | = | 99469.0 | nM | 4.00 |
| CHEMBL3193844 | — | IC50 | > | 118589.0 | nM | - |