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Assay Detail

CHEMBL1805702

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Competitive inhibition of CYP2C9
4
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Cytochrome P450 2C9 (CHEMBL3397)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of MK-0952, a selective PDE4 inhibitor for the treatment of long-term memory loss and mild cognitive impairment.
Gallant M, Aspiotis R, Day S, Dias R, Dubé D, Dubé L, Friesen RW, Girard M, Guay D, Hamel P, Huang Z, Lacombe P, Laliberté S, Lévesque JF, Liu S, Macdonald D, Mancini J, Nicholson DW, Styhler A, Townson K, Waters K, Young RN, Girard Y.
Bioorg Med Chem Lett (2010) 20 : 6387 -6393
PubMed 20933411 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 5.22 5.77

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL253083 2 5.77
CHEMBL485629 MK-0873 2.0 1 4.40
CHEMBL372575 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL253083 IC50 = 1700.0 nM 5.77
CHEMBL253083 IC50 = 3200.0 nM 5.50
CHEMBL485629 MK-0873 IC50 = 40000.0 nM 4.40
CHEMBL372575 IC50 < 1000.0 nM -