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Assay Detail

CHEMBL1832284

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Functional
Antiviral activity against Vaccinia virus infected in HEL cells assessed as inhibition of virus-induced cytopathic effect
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Vaccinia virus
Cell Type HEL
Confidence 1 — Organism
Curated By Autocuration

Target

Vaccinia virus (CHEMBL613493)
Type ORGANISM
Organism Vaccinia virus

Publication

Acyclic nucleoside thiophosphonates as potent inhibitors of HIV and HBV replication.
Barral K, Weck C, Payrot N, Roux L, Durafour C, Zoulim F, Neyts J, Balzarini J, Canard B, Priet S, Alvarez K.
Eur J Med Chem (2011) 46 : 4281 -4288
PubMed 21803462 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 4.09 4.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1830069 1 4.10
CHEMBL1830068 1 4.08
CHEMBL484 ADEFOVIR 3.0 1 -
CHEMBL483 TENOFOVIR ANHYDROUS 3.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1830069 EC50 = 80000.0 nM 4.10
CHEMBL1830068 EC50 = 84000.0 nM 4.08
CHEMBL484 ADEFOVIR EC50 > 200000.0 nM -
CHEMBL483 TENOFOVIR ANHYDROUS EC50 > 200000.0 nM -