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Assay Detail

CHEMBL1908641

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Binding
Binding constant for ALK kinase domain
72
Total Activities
72
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

ALK tyrosine kinase receptor (CHEMBL4247)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Comprehensive analysis of kinase inhibitor selectivity.
Davis MI, Hunt JP, Herrgard S, Ciceri P, Wodicka LM, Pallares G, Hocker M, Treiber DK, Zarrinkar PP.
Nat Biotechnol (2011) 29 : 1046 -1051
PubMed 22037378 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 72 6.48 9.26

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL464552 1 9.26
CHEMBL509032 TAE-684 1 8.96
CHEMBL601719 CRIZOTINIB 4.0 1 8.48
CHEMBL502835 NINTEDANIB 4.0 1 7.51
CHEMBL388978 STAUROSPORINE 1 7.50
CHEMBL1230609 FORETINIB 2.0 1 7.16
CHEMBL603469 LESTAURTINIB 3.0 1 7.15
CHEMBL513909 BI-2536 2.0 1 6.80
CHEMBL535 SUNITINIB 4.0 1 6.77
CHEMBL475251 R-406 2.0 1 6.62
CHEMBL608533 MIDOSTAURIN 4.0 1 6.57
CHEMBL1721885 SU-014813 2.0 1 6.31
CHEMBL1287853 FEDRATINIB 4.0 1 6.19
CHEMBL1908397 KW-2449 1.0 1 6.18
CHEMBL428690 ALVOCIDIB 3.0 1 6.17
CHEMBL288441 BOSUTINIB 4.0 1 6.16
CHEMBL1908395 1 6.08
CHEMBL1241674 1 5.96
CHEMBL553 ERLOTINIB 4.0 1 5.92
CHEMBL574738 AST-487 1.0 1 5.85
CHEMBL1789941 RUXOLITINIB 4.0 1 5.82
CHEMBL223360 LINIFANIB 3.0 1 5.80
CHEMBL24828 VANDETANIB 4.0 1 5.68
CHEMBL477772 PAZOPANIB 4.0 1 5.66
CHEMBL491473 CEDIRANIB 3.0 1 5.64
CHEMBL450786 PHA-665752 1 5.57
CHEMBL572878 TOZASERTIB 2.0 1 5.51
CHEMBL522892 DOVITINIB 3.0 1 5.46
CHEMBL31965 CANERTINIB 3.0 1 5.11
CHEMBL10 SB-203580 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL464552 Kd = 0.55 nM 9.26
CHEMBL509032 TAE-684 Kd = 1.1 nM 8.96
CHEMBL601719 CRIZOTINIB Kd = 3.3 nM 8.48
CHEMBL502835 NINTEDANIB Kd = 31.0 nM 7.51
CHEMBL388978 STAUROSPORINE Kd = 32.0 nM 7.50
CHEMBL1230609 FORETINIB Kd = 69.0 nM 7.16
CHEMBL603469 LESTAURTINIB Kd = 71.0 nM 7.15
CHEMBL513909 BI-2536 Kd = 160.0 nM 6.80
CHEMBL535 SUNITINIB Kd = 170.0 nM 6.77
CHEMBL475251 R-406 Kd = 240.0 nM 6.62
CHEMBL608533 MIDOSTAURIN Kd = 270.0 nM 6.57
CHEMBL1721885 SU-014813 Kd = 490.0 nM 6.31
CHEMBL1287853 FEDRATINIB Kd = 650.0 nM 6.19
CHEMBL1908397 KW-2449 Kd = 660.0 nM 6.18
CHEMBL428690 ALVOCIDIB Kd = 670.0 nM 6.17
CHEMBL288441 BOSUTINIB Kd = 690.0 nM 6.16
CHEMBL1908395 Kd = 840.0 nM 6.08
CHEMBL1241674 Kd = 1100.0 nM 5.96
CHEMBL553 ERLOTINIB Kd = 1200.0 nM 5.92
CHEMBL574738 AST-487 Kd = 1400.0 nM 5.85
CHEMBL1789941 RUXOLITINIB Kd = 1500.0 nM 5.82
CHEMBL223360 LINIFANIB Kd = 1600.0 nM 5.80
CHEMBL24828 VANDETANIB Kd = 2100.0 nM 5.68
CHEMBL477772 PAZOPANIB Kd = 2200.0 nM 5.66
CHEMBL491473 CEDIRANIB Kd = 2300.0 nM 5.64
CHEMBL450786 PHA-665752 Kd = 2700.0 nM 5.57
CHEMBL572878 TOZASERTIB Kd = 3100.0 nM 5.51
CHEMBL522892 DOVITINIB Kd = 3500.0 nM 5.46
CHEMBL31965 CANERTINIB Kd = 7700.0 nM 5.11
CHEMBL296468 BMS-387032 Kd > 10000.0 nM -
CHEMBL221959 TOFACITINIB Kd > 10000.0 nM -
CHEMBL180022 NERATINIB Kd > 10000.0 nM -
CHEMBL105442 CI-1040 Kd > 10000.0 nM -
CHEMBL215152 DEFOSBARASERTIB Kd > 10000.0 nM -
CHEMBL1336 SORAFENIB Kd > 10000.0 nM -
CHEMBL261849 GW632580X Kd > 10000.0 nM -
CHEMBL445813 AT-7519 Kd > 10000.0 nM -
CHEMBL255863 NILOTINIB Kd > 10000.0 nM -
CHEMBL494089 GSK-690693 Kd > 10000.0 nM -
CHEMBL558752 RAF-265 Kd > 10000.0 nM -
CHEMBL386051 Kd > 10000.0 nM -
CHEMBL1614701 SELUMETINIB Kd > 10000.0 nM -
CHEMBL259084 MLN-8054 Kd > 10000.0 nM -
CHEMBL1908394 GSK-461364 Kd > 10000.0 nM -
CHEMBL572881 MOTESANIB Kd > 10000.0 nM -
CHEMBL1236107 SGX-523 Kd > 10000.0 nM -
CHEMBL124660 TANDUTINIB Kd > 10000.0 nM -
CHEMBL941 IMATINIB Kd > 10000.0 nM -
CHEMBL939 GEFITINIB Kd > 10000.0 nM -
CHEMBL10 SB-203580 Kd > 10000.0 nM -