Assay Detail
Binding
CHEMBL1932156
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Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins
5
Total Activities
5
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Cannabinomimetic lipid from a marine cyanobacterium.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 8.02 | 8.02 |
| Ki | 2 | 8.68 | 8.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL188 | WIN-552122 | — | 1 | 8.68 |
| CHEMBL465 | DRONABINOL | 4.0 | 1 | 8.02 |
| CHEMBL1928586 | SERINOLAMIDE A | — | 1 | - |
| CHEMBL1928587 | — | — | 1 | - |
| CHEMBL1928588 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL188 | WIN-552122 | Ki | = | 2.1 | nM | 8.68 |
| CHEMBL465 | DRONABINOL | IC50 | = | 9.5 | nM | 8.02 |
| CHEMBL1928586 | SERINOLAMIDE A | IC50 | > | 10000.0 | nM | - |
| CHEMBL1928587 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1928588 | — | Ki | > | 10000.0 | nM | - |