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Assay Detail

CHEMBL1963719

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: DAPK3
ChEMBL ↗
945
Total Activities
927
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category other
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Death-associated protein kinase 3 (CHEMBL2468) ↗
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 945 6.34 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL21156 — — 1 9.00
CHEMBL1980995 — — 1 8.70
CHEMBL474432 — — 1 8.60
CHEMBL1998159 — — 1 8.40
CHEMBL1980407 — — 1 8.30
CHEMBL1984548 — — 1 8.30
CHEMBL1980329 — — 1 8.10
CHEMBL2000345 — — 1 8.10
CHEMBL1999931 — — 1 8.10
CHEMBL1980435 — — 1 7.90
CHEMBL1994669 — — 1 7.90
CHEMBL1998432 — — 1 7.90
CHEMBL1994241 — — 1 7.80
CHEMBL1969523 — — 1 7.80
CHEMBL2002613 — — 1 7.80
CHEMBL1970522 — — 1 7.80
CHEMBL1985723 — — 1 7.80
CHEMBL1997129 — — 1 7.70
CHEMBL1964399 — — 1 7.70
CHEMBL2005475 — — 1 7.70
CHEMBL2001751 — — 1 7.70
CHEMBL1983923 — — 1 7.70
CHEMBL1987261 — — 1 7.60
CHEMBL2000354 — — 1 7.60
CHEMBL1966343 — — 1 7.60
CHEMBL226403 — — 1 7.60
CHEMBL1968930 — — 1 7.60
CHEMBL1999484 — — 1 7.60
CHEMBL1987034 — — 1 7.50
CHEMBL523823 — — 1 7.50

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL21156 — Ki = 1.0 nM 9.00
CHEMBL1980995 — Ki = 1.995 nM 8.70
CHEMBL474432 — Ki = 2.512 nM 8.60
CHEMBL1998159 — Ki = 3.981 nM 8.40
CHEMBL1980407 — Ki = 5.012 nM 8.30
CHEMBL1984548 — Ki = 5.012 nM 8.30
CHEMBL1980329 — Ki = 7.943 nM 8.10
CHEMBL1999931 — Ki = 7.943 nM 8.10
CHEMBL2000345 — Ki = 7.943 nM 8.10
CHEMBL1980435 — Ki = 12.59 nM 7.90
CHEMBL1998432 — Ki = 12.59 nM 7.90
CHEMBL1994669 — Ki = 12.59 nM 7.90
CHEMBL2002613 — Ki = 15.85 nM 7.80
CHEMBL1970522 — Ki = 15.85 nM 7.80
CHEMBL1969523 — Ki = 15.85 nM 7.80
CHEMBL1994241 — Ki = 15.85 nM 7.80
CHEMBL1985723 — Ki = 15.85 nM 7.80
CHEMBL1983923 — Ki = 19.95 nM 7.70
CHEMBL2005475 — Ki = 19.95 nM 7.70
CHEMBL2001751 — Ki = 19.95 nM 7.70
CHEMBL1997129 — Ki = 19.95 nM 7.70
CHEMBL1964399 — Ki = 19.95 nM 7.70
CHEMBL1966343 — Ki = 25.12 nM 7.60
CHEMBL1999484 — Ki = 25.12 nM 7.60
CHEMBL226403 — Ki = 25.12 nM 7.60
CHEMBL1968930 — Ki = 25.12 nM 7.60
CHEMBL2000354 — Ki = 25.12 nM 7.60
CHEMBL1987261 — Ki = 25.12 nM 7.60
CHEMBL1987034 — Ki = 31.62 nM 7.50
CHEMBL1975128 — Ki = 31.62 nM 7.50
CHEMBL1991078 — Ki = 31.62 nM 7.50
CHEMBL523823 — Ki = 31.62 nM 7.50
CHEMBL1969537 — Ki = 31.62 nM 7.50
CHEMBL1975418 — Ki = 31.62 nM 7.50
CHEMBL1996980 — Ki = 31.62 nM 7.50
CHEMBL2005899 — Ki = 39.81 nM 7.40
CHEMBL1995813 — Ki = 39.81 nM 7.40
CHEMBL1966808 — Ki = 39.81 nM 7.40
CHEMBL1992363 — Ki = 39.81 nM 7.40
CHEMBL2000685 — Ki = 39.81 nM 7.40
CHEMBL1973098 — Ki = 39.81 nM 7.40
CHEMBL2005216 — Ki = 39.81 nM 7.40
CHEMBL1987448 — Ki = 39.81 nM 7.40
CHEMBL1973720 — Ki = 50.12 nM 7.30
CHEMBL2005718 — Ki = 50.12 nM 7.30
CHEMBL2003638 — Ki = 50.12 nM 7.30
CHEMBL1972339 — Ki = 50.12 nM 7.30
CHEMBL1966204 — Ki = 50.12 nM 7.30
CHEMBL1973720 — Ki = 50.12 nM 7.30
CHEMBL1995811 — Ki = 50.12 nM 7.30