| Serine/threonine-protein kinase pim-3 CHEMBL5407 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Serine/threonine-protein kinase pim-1 CHEMBL2147 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Serine/threonine-protein kinase pim-2 CHEMBL4523 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Death-associated protein kinase 3 CHEMBL2468 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Casein kinase II subunit alpha CHEMBL3629 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Tyrosine-protein kinase ABL1 CHEMBL1862 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Tyrosine-protein kinase Fyn CHEMBL1841 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Ribosomal protein S6 kinase alpha-3 CHEMBL2345 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta CHEMBL2801 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Proto-oncogene tyrosine-protein kinase ROS CHEMBL5568 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Homeodomain-interacting protein kinase 2 CHEMBL4576 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Serine/threonine-protein kinase PLK3 CHEMBL4897 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Ribosomal protein S6 kinase beta-1 CHEMBL4501 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| High affinity nerve growth factor receptor CHEMBL2815 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Serine/threonine-protein kinase PLK1 CHEMBL3024 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| SRSF protein kinase 1 CHEMBL4375 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Ribosomal protein S6 kinase alpha-5 CHEMBL4237 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Tyrosine-protein kinase Blk CHEMBL2250 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Homeodomain-interacting protein kinase 4 CHEMBL1075167 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma CHEMBL3829 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Tyrosine-protein kinase receptor TYRO3 CHEMBL5314 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Lymphokine-activated killer T-cell-originated protein kinase CHEMBL4896 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Interleukin-1 receptor-associated kinase 1 CHEMBL3357 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| MAP kinase-activated protein kinase 3 CHEMBL4670 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Serine/threonine-protein kinase Sgk2 CHEMBL5794 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Serine/threonine-protein kinase TAO1 CHEMBL5261 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Maternal embryonic leucine zipper kinase CHEMBL4578 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Serine/threonine-protein kinase Chk2 CHEMBL2527 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Mitogen-activated protein kinase kinase kinase 20 CHEMBL3886 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| MAP kinase-activated protein kinase 5 CHEMBL3094 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Serine/threonine-protein kinase Nek4 CHEMBL5819 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| MAP kinase-activated protein kinase 2 CHEMBL2208 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| RAC-alpha serine/threonine-protein kinase CHEMBL4282 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| Casein kinase I isoform gamma-3 CHEMBL5084 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| RAC-beta serine/threonine-protein kinase CHEMBL2431 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 5.4 | 5.4 | 3981.1 | 1 |