Assay Detail
Functional
CHEMBL1963754
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: HIPK2
693
Total Activities
680
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Homeodomain-interacting protein kinase 2 (CHEMBL4576) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 693 | 6.57 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1997554 | — | — | 1 | 8.40 |
| CHEMBL1983932 | — | — | 1 | 8.20 |
| CHEMBL243518 | — | — | 1 | 8.20 |
| CHEMBL243298 | — | — | 1 | 8.20 |
| CHEMBL1987448 | — | — | 1 | 8.20 |
| CHEMBL385478 | — | — | 1 | 8.20 |
| CHEMBL1967662 | — | — | 1 | 8.10 |
| CHEMBL1999931 | — | — | 1 | 8.10 |
| CHEMBL1996980 | — | — | 1 | 8.00 |
| CHEMBL1992363 | — | — | 1 | 7.90 |
| CHEMBL396523 | — | — | 1 | 7.90 |
| CHEMBL2003637 | — | — | 1 | 7.90 |
| CHEMBL1966628 | — | — | 1 | 7.80 |
| CHEMBL1964288 | — | — | 1 | 7.80 |
| CHEMBL213207 | — | — | 1 | 7.80 |
| CHEMBL1997643 | — | — | 1 | 7.70 |
| CHEMBL1241473 | — | — | 1 | 7.70 |
| CHEMBL1999153 | — | — | 1 | 7.70 |
| CHEMBL1974250 | — | — | 1 | 7.70 |
| CHEMBL1970821 | — | — | 1 | 7.60 |
| CHEMBL2005509 | — | — | 1 | 7.60 |
| CHEMBL1995813 | — | — | 1 | 7.60 |
| CHEMBL244378 | — | — | 1 | 7.60 |
| CHEMBL1965660 | — | — | 2 | 7.60 |
| CHEMBL1972290 | — | — | 1 | 7.60 |
| CHEMBL1991078 | — | — | 1 | 7.60 |
| CHEMBL1966204 | — | — | 1 | 7.60 |
| CHEMBL2003638 | — | — | 1 | 7.50 |
| CHEMBL1980435 | — | — | 1 | 7.50 |
| CHEMBL1986943 | — | — | 2 | 7.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1997554 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1987448 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL243298 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL385478 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1983932 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL243518 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1967662 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1999931 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1996980 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL396523 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1992363 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL2003637 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL213207 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1964288 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1966628 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1974250 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1997643 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1999153 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1241473 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1970821 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1991078 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL2005509 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1965660 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL244378 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1966204 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1965660 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1972290 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1995813 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1980435 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1986943 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1992220 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1982271 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL2003638 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1982400 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1986943 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL379975 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL2001751 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1966816 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1973720 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1987261 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1965836 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL2005718 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1982711 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1973720 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1979933 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1986263 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1990708 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1987948 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1983589 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1982660 | — | Ki | = | 50.12 | nM | 7.30 |