| Glycogen synthase kinase-3 alpha CHEMBL2850 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Casein kinase II subunit alpha CHEMBL3629 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Focal adhesion kinase 1 CHEMBL2695 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| MAP kinase-activated protein kinase 2 CHEMBL2208 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Insulin receptor CHEMBL1981 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Serine/threonine-protein kinase Nek4 CHEMBL5819 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Protein-tyrosine kinase 2-beta CHEMBL5469 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Tyrosine-protein kinase Blk CHEMBL2250 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Mitogen-activated protein kinase 8 CHEMBL2276 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Serine/threonine-protein kinase PLK1 CHEMBL3024 | Ki | 7.92 | 7.91 | 12.0 | 2 |
| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Serine/threonine-protein kinase PLK3 CHEMBL4897 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Macrophage colony-stimulating factor 1 receptor CHEMBL1844 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Tyrosine-protein kinase Fyn CHEMBL1841 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Mitogen-activated protein kinase 9 CHEMBL4179 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Cyclin-dependent kinase 2 CHEMBL301 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Tyrosine-protein kinase ITK/TSK CHEMBL2959 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Homeodomain-interacting protein kinase 2 CHEMBL4576 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Serine/threonine-protein kinase Nek2 CHEMBL3835 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Insulin-like growth factor 1 receptor CHEMBL1957 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret CHEMBL2041 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Tyrosine-protein kinase Lyn CHEMBL3905 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Tyrosine-protein kinase JAK2 CHEMBL2971 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Serine/threonine-protein kinase 3 CHEMBL4708 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Serine/threonine-protein kinase PAK 4 CHEMBL4482 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Proto-oncogene tyrosine-protein kinase Src CHEMBL267 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Tyrosine-protein kinase receptor UFO CHEMBL4895 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Maternal embryonic leucine zipper kinase CHEMBL4578 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Tyrosine-protein kinase Lck CHEMBL258 | Ki | 7.4 | 7.4 | 39.8 | 1 |