Assay Detail
Functional
CHEMBL1963771
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: GSK3A
968
Total Activities
951
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 968 | 6.21 | 8.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1980407 | — | — | 1 | 8.90 |
| CHEMBL1241473 | — | — | 1 | 8.50 |
| CHEMBL2005936 | — | — | 1 | 8.40 |
| CHEMBL1973540 | — | — | 1 | 8.40 |
| CHEMBL396523 | — | — | 1 | 8.40 |
| CHEMBL1994830 | — | — | 1 | 8.40 |
| CHEMBL1995811 | — | — | 1 | 8.40 |
| CHEMBL1987430 | — | — | 1 | 8.30 |
| CHEMBL1975647 | — | — | 1 | 8.30 |
| CHEMBL1973483 | — | — | 1 | 8.30 |
| CHEMBL336961 | AZAKENPAULLONE | — | 1 | 8.30 |
| CHEMBL1999718 | — | — | 1 | 8.20 |
| CHEMBL1988153 | — | — | 1 | 8.20 |
| CHEMBL1994538 | — | — | 1 | 8.20 |
| CHEMBL1965660 | — | — | 2 | 8.20 |
| CHEMBL1992732 | — | — | 1 | 8.20 |
| CHEMBL1980435 | — | — | 1 | 8.20 |
| CHEMBL1984548 | — | — | 1 | 8.10 |
| CHEMBL296586 | KENPAULLONE | — | 1 | 8.10 |
| CHEMBL243088 | — | — | 1 | 8.10 |
| CHEMBL412142 | LADUVIGLUSIB | 1.0 | 1 | 8.00 |
| CHEMBL1986499 | — | — | 1 | 8.00 |
| CHEMBL1972119 | — | — | 1 | 8.00 |
| CHEMBL2002599 | — | — | 1 | 8.00 |
| CHEMBL2001987 | — | — | 1 | 7.90 |
| CHEMBL1994669 | — | — | 1 | 7.90 |
| CHEMBL2002613 | — | — | 1 | 7.90 |
| CHEMBL1972158 | — | — | 1 | 7.80 |
| CHEMBL1981215 | — | — | 1 | 7.80 |
| CHEMBL1966703 | — | — | 1 | 7.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1980407 | — | Ki | = | 1.259 | nM | 8.90 |
| CHEMBL1241473 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1973540 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL396523 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL2005936 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1995811 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1994830 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1973483 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1975647 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1987430 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL336961 | AZAKENPAULLONE | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1980435 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1994538 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1965660 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1992732 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1965660 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1988153 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1999718 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL296586 | KENPAULLONE | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL243088 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1984548 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL2002599 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL412142 | LADUVIGLUSIB | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1972119 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1986499 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1994669 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL2001987 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL2002613 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL2000104 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1981744 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1975418 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1972158 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1981215 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1966703 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL242865 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1980995 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1967564 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL243298 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1682553 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1980142 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1997534 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1975787 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1967336 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL526133 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL259850 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL497151 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1966524 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1968070 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1999918 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL2003817 | — | Ki | = | 25.12 | nM | 7.60 |