| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Glycogen synthase kinase-3 alpha CHEMBL2850 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Serine/threonine-protein kinase 17A CHEMBL4525 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Serine/threonine-protein kinase N2 CHEMBL3032 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Maternal embryonic leucine zipper kinase CHEMBL4578 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret CHEMBL2041 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Fibroblast growth factor receptor 3 CHEMBL2742 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Serine/threonine-protein kinase BRSK1 CHEMBL5650 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 CHEMBL2534 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Serine/threonine-protein kinase Sgk2 CHEMBL5794 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| High affinity nerve growth factor receptor CHEMBL2815 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Interleukin-1 receptor-associated kinase 1 CHEMBL3357 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Tyrosine-protein kinase receptor UFO CHEMBL4895 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Tyrosine-protein kinase JAK3 CHEMBL2148 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Tyrosine-protein kinase FRK CHEMBL4223 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Ribosomal protein S6 kinase alpha-3 CHEMBL2345 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Rho-associated protein kinase 2 CHEMBL2973 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Death-associated protein kinase 3 CHEMBL2468 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta CHEMBL2801 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Casein kinase I isoform delta CHEMBL2828 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| BDNF/NT-3 growth factors receptor CHEMBL4898 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Tyrosine-protein kinase BTK CHEMBL5251 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Mitogen-activated protein kinase 8 CHEMBL2276 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Tyrosine-protein kinase Lck CHEMBL258 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Tyrosine-protein kinase ITK/TSK CHEMBL2959 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Mitogen-activated protein kinase 9 CHEMBL4179 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| cGMP-dependent protein kinase 1 CHEMBL4273 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Ribosomal protein S6 kinase beta-1 CHEMBL4501 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Homeodomain-interacting protein kinase 2 CHEMBL4576 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Tyrosine-protein kinase receptor TYRO3 CHEMBL5314 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 6.9 | 6.9 | 125.9 | 1 |