Assay Detail
Functional
CHEMBL1963727
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: STK6
951
Total Activities
938
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 951 | 6.53 | 9.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL483158 | ALISERTIB | 3.0 | 1 | 9.30 |
| CHEMBL1972576 | — | — | 1 | 9.20 |
| CHEMBL1987034 | — | — | 1 | 8.80 |
| CHEMBL1972220 | — | — | 1 | 8.80 |
| CHEMBL2002165 | — | — | 1 | 8.70 |
| CHEMBL1965170 | — | — | 1 | 8.70 |
| CHEMBL1979516 | — | — | 1 | 8.70 |
| CHEMBL1980297 | ILORASERTIB | 2.0 | 1 | 8.70 |
| CHEMBL1980995 | — | — | 1 | 8.60 |
| CHEMBL1970203 | — | — | 1 | 8.60 |
| CHEMBL244793 | — | — | 1 | 8.60 |
| CHEMBL1982476 | — | — | 1 | 8.50 |
| CHEMBL572878 | TOZASERTIB | 2.0 | 1 | 8.50 |
| CHEMBL1967720 | — | — | 1 | 8.50 |
| CHEMBL1967878 | CENISERTIB | 2.0 | 1 | 8.40 |
| CHEMBL1989708 | — | — | 2 | 8.40 |
| CHEMBL1970317 | — | — | 1 | 8.40 |
| CHEMBL1983111 | — | — | 1 | 8.40 |
| CHEMBL1972851 | — | — | 1 | 8.40 |
| CHEMBL1967531 | — | — | 1 | 8.30 |
| CHEMBL243749 | — | — | 1 | 8.30 |
| CHEMBL1993661 | — | — | 1 | 8.30 |
| CHEMBL1993941 | — | — | 1 | 8.20 |
| CHEMBL1967116 | — | — | 1 | 8.20 |
| CHEMBL243517 | — | — | 1 | 8.20 |
| CHEMBL2004290 | — | — | 1 | 8.20 |
| CHEMBL2005631 | — | — | 1 | 8.20 |
| CHEMBL1980144 | — | — | 1 | 8.20 |
| CHEMBL1970142 | — | — | 1 | 8.10 |
| CHEMBL1990228 | — | — | 1 | 8.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL483158 | ALISERTIB | Ki | = | 0.5012 | nM | 9.30 |
| CHEMBL1972576 | — | Ki | = | 0.631 | nM | 9.20 |
| CHEMBL1987034 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL1972220 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL1965170 | — | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL1980297 | ILORASERTIB | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL2002165 | — | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL1979516 | — | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL1970203 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL1980995 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL244793 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL572878 | TOZASERTIB | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1982476 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1967720 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1972851 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1983111 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1970317 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1967878 | CENISERTIB | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1989708 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL243749 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1993661 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1967531 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1967116 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL2004290 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1980144 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1989708 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL2005631 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL243517 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1993941 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1987054 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1981047 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1990228 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1972584 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1970142 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL2000393 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1974254 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1982466 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL2006715 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1965570 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1977041 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL243088 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL2004716 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL509032 | TAE-684 | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1983923 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1973540 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL243518 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL2007064 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1988437 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1978099 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1964519 | — | Ki | = | 19.95 | nM | 7.70 |