| Leucine-rich repeat serine/threonine-protein kinase 2 CHEMBL1075104 | Ki | 9.2 | 9.2 | 0.6 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret CHEMBL2041 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Tyrosine-protein kinase Fer CHEMBL3982 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Serine/threonine-protein kinase 17A CHEMBL4525 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Tyrosine-protein kinase ITK/TSK CHEMBL2959 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Tyrosine-protein kinase JAK2 CHEMBL2971 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Fibroblast growth factor receptor 3 CHEMBL2742 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Focal adhesion kinase 1 CHEMBL2695 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Ribosomal protein S6 kinase alpha-3 CHEMBL2345 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Non-receptor tyrosine-protein kinase TYK2 CHEMBL3553 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Serine/threonine-protein kinase TBK1 CHEMBL5408 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Tyrosine-protein kinase Fes/Fps CHEMBL5455 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 CHEMBL2534 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Cyclin-dependent kinase 2 CHEMBL301 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Serine/threonine-protein kinase Chk1 CHEMBL4630 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Macrophage-stimulating protein receptor CHEMBL2689 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Insulin receptor CHEMBL1981 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Tyrosine-protein kinase JAK3 CHEMBL2148 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 CHEMBL4852 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Tyrosine-protein kinase SYK CHEMBL2599 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| BDNF/NT-3 growth factors receptor CHEMBL4898 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Proto-oncogene tyrosine-protein kinase ROS CHEMBL5568 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit epsilon CHEMBL3529 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| NT-3 growth factor receptor CHEMBL5608 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Leukocyte tyrosine kinase receptor CHEMBL5627 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Insulin-like growth factor 1 receptor CHEMBL1957 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Serine/threonine-protein kinase Chk2 CHEMBL2527 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Serine/threonine-protein kinase 3 CHEMBL4708 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Testis-specific serine/threonine-protein kinase 1 CHEMBL6003 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Macrophage colony-stimulating factor 1 receptor CHEMBL1844 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Platelet-derived growth factor receptor beta CHEMBL1913 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Proto-oncogene tyrosine-protein kinase Src CHEMBL267 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Interleukin-1 receptor-associated kinase 1 CHEMBL3357 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Activated CDC42 kinase 1 CHEMBL4599 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Serine/threonine-protein kinase D3 CHEMBL2595 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Tyrosine-protein kinase FRK CHEMBL4223 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Serine/threonine-protein kinase BRSK1 CHEMBL5650 | Ki | 7.1 | 7.1 | 79.4 | 1 |