Assay Detail
Functional
CHEMBL1963806
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: LRRK2
346
Total Activities
336
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Leucine-rich repeat serine/threonine-protein kinase 2 (CHEMBL1075104) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 346 | 6.26 | 9.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1993661 | — | — | 1 | 9.50 |
| CHEMBL1980995 | — | — | 1 | 9.40 |
| CHEMBL1967878 | CENISERTIB | 2.0 | 1 | 9.20 |
| CHEMBL1983111 | — | — | 1 | 9.20 |
| CHEMBL2006765 | — | — | 1 | 9.10 |
| CHEMBL2006564 | — | — | 1 | 8.90 |
| CHEMBL1973720 | — | — | 2 | 8.70 |
| CHEMBL458997 | — | — | 1 | 8.60 |
| CHEMBL1980407 | — | — | 1 | 8.20 |
| CHEMBL461876 | — | — | 1 | 8.10 |
| CHEMBL1986943 | — | — | 2 | 8.10 |
| CHEMBL1980329 | — | — | 1 | 8.10 |
| CHEMBL1997924 | — | — | 1 | 8.00 |
| CHEMBL1974328 | — | — | 1 | 7.90 |
| CHEMBL1979690 | — | — | 1 | 7.80 |
| CHEMBL1977138 | — | — | 1 | 7.80 |
| CHEMBL1969151 | — | — | 1 | 7.80 |
| CHEMBL2004118 | — | — | 1 | 7.80 |
| CHEMBL1983715 | — | — | 1 | 7.70 |
| CHEMBL2002992 | — | — | 1 | 7.70 |
| CHEMBL1998953 | — | — | 1 | 7.70 |
| CHEMBL1988437 | — | — | 1 | 7.70 |
| CHEMBL1980763 | — | — | 1 | 7.60 |
| CHEMBL1972220 | — | — | 1 | 7.60 |
| CHEMBL1980297 | ILORASERTIB | 2.0 | 1 | 7.60 |
| CHEMBL1975927 | — | — | 1 | 7.60 |
| CHEMBL21156 | — | — | 1 | 7.60 |
| CHEMBL1967998 | — | — | 1 | 7.50 |
| CHEMBL475251 | R-406 | 2.0 | 1 | 7.50 |
| CHEMBL1991674 | — | — | 1 | 7.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1993661 | — | Ki | = | 0.3162 | nM | 9.50 |
| CHEMBL1980995 | — | Ki | = | 0.3981 | nM | 9.40 |
| CHEMBL1983111 | — | Ki | = | 0.631 | nM | 9.20 |
| CHEMBL1967878 | CENISERTIB | Ki | = | 0.631 | nM | 9.20 |
| CHEMBL2006765 | — | Ki | = | 0.7943 | nM | 9.10 |
| CHEMBL2006564 | — | Ki | = | 1.259 | nM | 8.90 |
| CHEMBL1973720 | — | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL1973720 | — | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL458997 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL1980407 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1986943 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL461876 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1980329 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1986943 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1997924 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1974328 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1977138 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1969151 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL2004118 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1979690 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1998953 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1988437 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL2002992 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1983715 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1980297 | ILORASERTIB | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL21156 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1980763 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1975927 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1972220 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1997007 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL475251 | R-406 | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1991674 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL2002586 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1967998 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL2000029 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL2007559 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1983348 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1984760 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1999484 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1983575 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL1989708 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL235157 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL1081312 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL2002099 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1973516 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL2007574 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL191003 | JNJ-7706621 | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1988581 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL379975 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL1982753 | — | Ki | = | 100.0 | nM | 7.00 |