| Tyrosine-protein kinase JAK2 CHEMBL2971 | Ki | 8.6 | 8.6 | 2.5 | 1 |
| Wee1-like protein kinase CHEMBL5491 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Macrophage colony-stimulating factor 1 receptor CHEMBL1844 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret CHEMBL2041 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Insulin-like growth factor 1 receptor CHEMBL1957 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Serine/threonine-protein kinase TAO1 CHEMBL5261 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Leukocyte tyrosine kinase receptor CHEMBL5627 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Leucine-rich repeat serine/threonine-protein kinase 2 CHEMBL1075104 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Tyrosine-protein kinase Lck CHEMBL258 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Mitogen-activated protein kinase 8 CHEMBL2276 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Serine/threonine-protein kinase D3 CHEMBL2595 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Tyrosine-protein kinase JAK3 CHEMBL2148 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Activated CDC42 kinase 1 CHEMBL4599 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Cyclin-dependent kinase 7 CHEMBL3055 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Focal adhesion kinase 1 CHEMBL2695 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Mitogen-activated protein kinase 9 CHEMBL4179 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha CHEMBL4101 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| ALK tyrosine kinase receptor CHEMBL4247 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 2 CHEMBL2964 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Serine/threonine-protein kinase PAK 4 CHEMBL4482 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 1 CHEMBL3587 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Activin receptor type-1 CHEMBL5903 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Ribosomal protein S6 kinase alpha-3 CHEMBL2345 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Platelet-derived growth factor receptor alpha CHEMBL2007 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B CHEMBL5543 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| BDNF/NT-3 growth factors receptor CHEMBL4898 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Tyrosine-protein kinase Fyn CHEMBL1841 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Death-associated protein kinase 3 CHEMBL2468 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Tyrosine-protein kinase receptor TYRO3 CHEMBL5314 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| High affinity nerve growth factor receptor CHEMBL2815 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Rho-associated protein kinase 1 CHEMBL3231 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Serine/threonine-protein kinase TBK1 CHEMBL5408 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Tyrosine-protein kinase BTK CHEMBL5251 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| NT-3 growth factor receptor CHEMBL5608 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Macrophage-stimulating protein receptor CHEMBL2689 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Cyclin-dependent kinase 9 CHEMBL3116 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| cAMP-dependent protein kinase catalytic subunit PRKX CHEMBL5818 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Cyclin-dependent kinase 19 CHEMBL6002 | Ki | 6.0 | 6.0 | 1000.0 | 1 |