Assay Detail
Functional
CHEMBL1963718
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: LCK
952
Total Activities
934
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 952 | 6.46 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1988387 | — | — | 1 | 9.00 |
| CHEMBL1967116 | — | — | 1 | 9.00 |
| CHEMBL1970142 | — | — | 1 | 9.00 |
| CHEMBL49120 | PD-0166285 | 1.0 | 1 | 8.90 |
| CHEMBL1972220 | — | — | 1 | 8.90 |
| CHEMBL1965170 | — | — | 1 | 8.80 |
| CHEMBL1988717 | — | — | 1 | 8.80 |
| CHEMBL1970317 | — | — | 1 | 8.80 |
| CHEMBL1974254 | — | — | 1 | 8.80 |
| CHEMBL1981725 | — | — | 1 | 8.70 |
| CHEMBL1980297 | ILORASERTIB | 2.0 | 1 | 8.70 |
| CHEMBL2006715 | — | — | 1 | 8.60 |
| CHEMBL1976376 | — | — | 1 | 8.60 |
| CHEMBL1967720 | — | — | 1 | 8.60 |
| CHEMBL2002165 | — | — | 1 | 8.50 |
| CHEMBL2001485 | — | — | 1 | 8.40 |
| CHEMBL2004290 | — | — | 1 | 8.40 |
| CHEMBL1989708 | — | — | 1 | 8.40 |
| CHEMBL1967878 | CENISERTIB | 2.0 | 1 | 8.20 |
| CHEMBL2005631 | — | — | 1 | 8.20 |
| CHEMBL1989267 | — | — | 1 | 8.10 |
| CHEMBL1986851 | — | — | 1 | 8.10 |
| CHEMBL1984711 | — | — | 1 | 8.10 |
| CHEMBL1979516 | — | — | 1 | 8.10 |
| CHEMBL1991429 | — | — | 1 | 8.00 |
| CHEMBL2004716 | — | — | 1 | 8.00 |
| CHEMBL1984162 | — | — | 1 | 8.00 |
| CHEMBL1996979 | — | — | 1 | 7.90 |
| CHEMBL1982476 | — | — | 1 | 7.90 |
| CHEMBL574738 | AST-487 | 1.0 | 1 | 7.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1988387 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL1967116 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL1970142 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL49120 | PD-0166285 | Ki | = | 1.259 | nM | 8.90 |
| CHEMBL1972220 | — | Ki | = | 1.259 | nM | 8.90 |
| CHEMBL1988717 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL1974254 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL1970317 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL1965170 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL1980297 | ILORASERTIB | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL1981725 | — | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL1976376 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL2006715 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL1967720 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL2002165 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL2004290 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1989708 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL2001485 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL2005631 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1967878 | CENISERTIB | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1986851 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1989267 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1984711 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1979516 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL2004716 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1991429 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1984162 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1982476 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1996979 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL574738 | AST-487 | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1994938 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1965570 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL522892 | DOVITINIB | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1090360 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1966514 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1980995 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1970083 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1979690 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1969102 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1973178 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1967998 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1983923 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1977134 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1999414 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1990885 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1996649 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1241473 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL2001228 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL273187 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1090356 | — | Ki | = | 39.81 | nM | 7.40 |