Assay Detail
Functional
CHEMBL1963792
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: IGF1R
814
Total Activities
801
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Insulin-like growth factor 1 receptor (CHEMBL1957) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 814 | 6.36 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2000271 | — | — | 1 | 9.00 |
| CHEMBL461876 | — | — | 1 | 8.70 |
| CHEMBL1991429 | — | — | 1 | 8.40 |
| CHEMBL458997 | — | — | 1 | 8.40 |
| CHEMBL1999811 | — | — | 1 | 8.30 |
| CHEMBL1993661 | — | — | 1 | 8.30 |
| CHEMBL1971029 | — | — | 1 | 8.20 |
| CHEMBL1090360 | — | — | 1 | 8.00 |
| CHEMBL1981725 | — | — | 1 | 7.90 |
| CHEMBL1979690 | — | — | 1 | 7.80 |
| CHEMBL1967998 | — | — | 1 | 7.70 |
| CHEMBL1984162 | — | — | 1 | 7.60 |
| CHEMBL1090356 | — | — | 1 | 7.60 |
| CHEMBL1241473 | — | — | 1 | 7.60 |
| CHEMBL1980995 | — | — | 1 | 7.60 |
| CHEMBL1966842 | — | — | 1 | 7.60 |
| CHEMBL1988163 | — | — | 1 | 7.60 |
| CHEMBL2005886 | — | — | 1 | 7.60 |
| CHEMBL1987034 | — | — | 1 | 7.50 |
| CHEMBL1996234 | — | — | 1 | 7.50 |
| CHEMBL1983111 | — | — | 1 | 7.30 |
| CHEMBL1983268 | ENTRECTINIB | 4.0 | 1 | 7.20 |
| CHEMBL1973516 | — | — | 2 | 7.10 |
| CHEMBL1997924 | — | — | 1 | 7.10 |
| CHEMBL2006715 | — | — | 1 | 7.10 |
| CHEMBL1968791 | — | — | 1 | 7.00 |
| CHEMBL1989708 | — | — | 1 | 7.00 |
| CHEMBL1991138 | — | — | 1 | 7.00 |
| CHEMBL2000078 | — | — | 1 | 6.80 |
| CHEMBL243088 | — | — | 1 | 6.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2000271 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL461876 | — | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL458997 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1991429 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1993661 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1999811 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1971029 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1090360 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1981725 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1979690 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1967998 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1980995 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1966842 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1988163 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1984162 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1241473 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL2005886 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1090356 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1987034 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1996234 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1983111 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1983268 | ENTRECTINIB | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL2006715 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1973516 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1997924 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1968791 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL1991138 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL1989708 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL1973516 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL243088 | — | Ki | = | 158.49 | nM | 6.80 |
| CHEMBL2000078 | — | Ki | = | 158.49 | nM | 6.80 |
| CHEMBL2005482 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1825138 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1974328 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1997909 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1988370 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1980297 | ILORASERTIB | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1984711 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL2006564 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1825138 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1987054 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1983715 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1999484 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1988581 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL101311 | — | Ki | = | 316.23 | nM | 6.50 |
| CHEMBL396523 | — | Ki | = | 316.23 | nM | 6.50 |
| CHEMBL1992323 | — | Ki | = | 316.23 | nM | 6.50 |
| CHEMBL1965910 | — | Ki | = | 398.11 | nM | 6.40 |
| CHEMBL1969102 | — | Ki | = | 398.11 | nM | 6.40 |
| CHEMBL1988141 | — | Ki | = | 398.11 | nM | 6.40 |