| ALK tyrosine kinase receptor CHEMBL4247 | Ki | 8.8 | 8.8 | 1.6 | 1 |
| Protein-tyrosine kinase 2-beta CHEMBL5469 | Ki | 8.8 | 8.8 | 1.6 | 1 |
| Testis-specific serine/threonine-protein kinase 1 CHEMBL6003 | Ki | 8.6 | 8.6 | 2.5 | 1 |
| Focal adhesion kinase 1 CHEMBL2695 | Ki | 8.6 | 8.6 | 2.5 | 1 |
| Tyrosine-protein kinase JAK2 CHEMBL2971 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Insulin-like growth factor 1 receptor CHEMBL1957 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Serine/threonine-protein kinase D3 CHEMBL2595 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Serine/threonine-protein kinase 3 CHEMBL4708 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Testis-specific serine/threonine-protein kinase 2 CHEMBL6014 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Tyrosine-protein kinase JAK3 CHEMBL2148 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Serine/threonine-protein kinase PAK 4 CHEMBL4482 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret CHEMBL2041 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Tyrosine-protein kinase Fyn CHEMBL1841 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Interleukin-1 receptor-associated kinase 1 CHEMBL3357 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Tyrosine-protein kinase receptor UFO CHEMBL4895 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Tyrosine-protein kinase ITK/TSK CHEMBL2959 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Serine/threonine-protein kinase TAO1 CHEMBL5261 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Tyrosine-protein kinase Blk CHEMBL2250 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Mast/stem cell growth factor receptor Kit CHEMBL1936 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Non-receptor tyrosine-protein kinase TYK2 CHEMBL3553 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Proto-oncogene tyrosine-protein kinase Src CHEMBL267 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Fibroblast growth factor receptor 3 CHEMBL2742 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Epidermal growth factor receptor CHEMBL203 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Tyrosine-protein kinase Lck CHEMBL258 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 CHEMBL4852 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Cyclin-dependent kinase 2 CHEMBL301 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Tyrosine-protein kinase Lyn CHEMBL3905 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Mitogen-activated protein kinase 1 CHEMBL4040 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 CHEMBL2534 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Serine/threonine-protein kinase N2 CHEMBL3032 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Macrophage colony-stimulating factor 1 receptor CHEMBL1844 | Ki | 6.8 | 6.8 | 158.5 | 1 |