Assay Detail
Functional
CHEMBL1964101
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: MAP4K4
1003
Total Activities
985
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Mitogen-activated protein kinase kinase kinase kinase 4 (CHEMBL6166) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1003 | 6.14 | 8.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1980995 | — | — | 1 | 8.80 |
| CHEMBL2006778 | — | — | 1 | 8.50 |
| CHEMBL1993648 | — | — | 1 | 8.50 |
| CHEMBL1970821 | — | — | 1 | 8.50 |
| CHEMBL1988331 | — | — | 1 | 8.40 |
| CHEMBL2001751 | — | — | 1 | 8.40 |
| CHEMBL385478 | — | — | 1 | 8.40 |
| CHEMBL1989006 | — | — | 1 | 8.40 |
| CHEMBL1980407 | — | — | 1 | 8.30 |
| CHEMBL1996980 | — | — | 1 | 8.20 |
| CHEMBL1965836 | — | — | 1 | 8.20 |
| CHEMBL1992220 | — | — | 1 | 8.20 |
| CHEMBL2002726 | — | — | 1 | 8.20 |
| CHEMBL1992634 | — | — | 1 | 8.10 |
| CHEMBL1986855 | — | — | 1 | 8.10 |
| CHEMBL1998068 | — | — | 1 | 8.00 |
| CHEMBL1983932 | — | — | 1 | 8.00 |
| CHEMBL1976936 | — | — | 1 | 8.00 |
| CHEMBL1983589 | — | — | 1 | 7.90 |
| CHEMBL2007002 | — | — | 1 | 7.90 |
| CHEMBL1982271 | — | — | 1 | 7.90 |
| CHEMBL2005509 | — | — | 1 | 7.90 |
| CHEMBL1968459 | — | — | 1 | 7.80 |
| CHEMBL1999279 | — | — | 1 | 7.80 |
| CHEMBL1241473 | — | — | 1 | 7.80 |
| CHEMBL2005216 | — | — | 1 | 7.80 |
| CHEMBL1971029 | — | — | 1 | 7.80 |
| CHEMBL1966816 | — | — | 1 | 7.70 |
| CHEMBL1980253 | — | — | 1 | 7.70 |
| CHEMBL213207 | — | — | 1 | 7.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1980995 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL2006778 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1970821 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1993648 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1988331 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL2001751 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL385478 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1989006 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1980407 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1965836 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1996980 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL2002726 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1992220 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1986855 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1992634 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1983932 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1998068 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1976936 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL2005509 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL2007002 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1983589 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1982271 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1971029 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1999279 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1968459 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1241473 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL2005216 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1973720 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1980253 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1999931 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1973720 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1966816 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1980329 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1985654 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1999153 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1967887 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL213207 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL363648 | TAK-715 | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1994938 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1997554 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL226471 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL522892 | DOVITINIB | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL2005718 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1972220 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1965507 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1998432 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1965423 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1966040 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1995813 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1970142 | — | Ki | = | 31.62 | nM | 7.50 |