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Assay Detail

CHEMBL1963691

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CLK2
ChEMBL ↗
910
Total Activities
893
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category other
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Dual specificity protein kinase CLK2 (CHEMBL4225) ↗
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 910 6.13 9.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1980407 — — 1 9.10
CHEMBL1981133 — — 1 8.60
CHEMBL1970903 — — 1 8.50
CHEMBL1996980 — — 1 8.50
CHEMBL1987448 — — 1 8.40
CHEMBL1969588 — — 1 8.40
CHEMBL1994669 — — 1 8.40
CHEMBL1986263 — — 1 8.30
CHEMBL1977138 — — 1 8.30
CHEMBL1967302 — — 1 8.30
CHEMBL1987679 — — 1 8.30
CHEMBL1966628 — — 1 8.30
CHEMBL1982711 — — 1 8.20
CHEMBL1973720 — — 2 8.10
CHEMBL1986943 — — 2 8.10
CHEMBL1982271 — — 1 8.00
CHEMBL1967887 — — 1 8.00
CHEMBL1984548 — — 1 8.00
CHEMBL1999931 — — 1 8.00
CHEMBL1682552 — — 1 7.90
CHEMBL1996817 — — 1 7.90
CHEMBL1992220 — — 1 7.80
CHEMBL1983575 — — 1 7.80
CHEMBL1987948 — — 1 7.80
CHEMBL2003638 — — 1 7.80
CHEMBL2005509 — — 1 7.80
CHEMBL1986855 — — 1 7.80
CHEMBL1987034 — — 1 7.80
CHEMBL1980253 — — 1 7.80
CHEMBL2007574 — — 1 7.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1980407 — Ki = 0.7943 nM 9.10
CHEMBL1981133 — Ki = 2.512 nM 8.60
CHEMBL1996980 — Ki = 3.162 nM 8.50
CHEMBL1970903 — Ki = 3.162 nM 8.50
CHEMBL1969588 — Ki = 3.981 nM 8.40
CHEMBL1994669 — Ki = 3.981 nM 8.40
CHEMBL1987448 — Ki = 3.981 nM 8.40
CHEMBL1986263 — Ki = 5.012 nM 8.30
CHEMBL1966628 — Ki = 5.012 nM 8.30
CHEMBL1987679 — Ki = 5.012 nM 8.30
CHEMBL1977138 — Ki = 5.012 nM 8.30
CHEMBL1967302 — Ki = 5.012 nM 8.30
CHEMBL1982711 — Ki = 6.31 nM 8.20
CHEMBL1973720 — Ki = 7.943 nM 8.10
CHEMBL1973720 — Ki = 7.943 nM 8.10
CHEMBL1986943 — Ki = 7.943 nM 8.10
CHEMBL1986943 — Ki = 7.943 nM 8.10
CHEMBL1982271 — Ki = 10.0 nM 8.00
CHEMBL1967887 — Ki = 10.0 nM 8.00
CHEMBL1999931 — Ki = 10.0 nM 8.00
CHEMBL1984548 — Ki = 10.0 nM 8.00
CHEMBL1996817 — Ki = 12.59 nM 7.90
CHEMBL1682552 — Ki = 12.59 nM 7.90
CHEMBL1980253 — Ki = 15.85 nM 7.80
CHEMBL1986855 — Ki = 15.85 nM 7.80
CHEMBL2003638 — Ki = 15.85 nM 7.80
CHEMBL1987948 — Ki = 15.85 nM 7.80
CHEMBL1983575 — Ki = 15.85 nM 7.80
CHEMBL1992220 — Ki = 15.85 nM 7.80
CHEMBL1998432 — Ki = 15.85 nM 7.80
CHEMBL2007574 — Ki = 15.85 nM 7.80
CHEMBL2005509 — Ki = 15.85 nM 7.80
CHEMBL1987034 — Ki = 15.85 nM 7.80
CHEMBL1980995 — Ki = 19.95 nM 7.70
CHEMBL1971029 — Ki = 19.95 nM 7.70
CHEMBL1998121 — Ki = 19.95 nM 7.70
CHEMBL1972290 — Ki = 19.95 nM 7.70
CHEMBL509032 TAE-684 Ki = 25.12 nM 7.60
CHEMBL1997129 — Ki = 25.12 nM 7.60
CHEMBL1987261 — Ki = 25.12 nM 7.60
CHEMBL1974935 — Ki = 25.12 nM 7.60
CHEMBL1966204 — Ki = 25.12 nM 7.60
CHEMBL1241473 — Ki = 31.62 nM 7.50
CHEMBL2002613 — Ki = 31.62 nM 7.50
CHEMBL1980562 — Ki = 31.62 nM 7.50
CHEMBL1971172 — Ki = 31.62 nM 7.50
CHEMBL1985723 — Ki = 31.62 nM 7.50
CHEMBL461876 — Ki = 31.62 nM 7.50
CHEMBL1980435 — Ki = 31.62 nM 7.50
CHEMBL2005718 — Ki = 39.81 nM 7.40