| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Rho-associated protein kinase 2 CHEMBL2973 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| RAC-alpha serine/threonine-protein kinase CHEMBL4282 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Serine/threonine-protein kinase N2 CHEMBL3032 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| cAMP-dependent protein kinase catalytic subunit PRKX CHEMBL5818 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Rho-associated protein kinase 1 CHEMBL3231 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| cGMP-dependent protein kinase 1 CHEMBL4273 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha CHEMBL4101 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| cGMP-dependent protein kinase 2 CHEMBL2896 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| RAC-beta serine/threonine-protein kinase CHEMBL2431 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Ribosomal protein S6 kinase alpha-5 CHEMBL4237 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Serine/threonine-protein kinase 17A CHEMBL4525 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 3 CHEMBL4575 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| RAC-gamma serine/threonine-protein kinase CHEMBL4816 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Glycogen synthase kinase-3 alpha CHEMBL2850 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Serine/threonine-protein kinase pim-1 CHEMBL2147 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Lymphokine-activated killer T-cell-originated protein kinase CHEMBL4896 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Protein kinase C delta type CHEMBL2996 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Ribosomal protein S6 kinase beta-1 CHEMBL4501 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha CHEMBL3476 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Serine/threonine-protein kinase D3 CHEMBL2595 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Ribosomal protein S6 kinase alpha-3 CHEMBL2345 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Serine/threonine-protein kinase pim-3 CHEMBL5407 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Protein kinase C gamma type CHEMBL2938 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Serine/threonine-protein kinase pim-2 CHEMBL4523 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Serine/threonine-protein kinase TAO1 CHEMBL5261 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Casein kinase I isoform gamma-2 CHEMBL2543 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Casein kinase I isoform gamma-1 CHEMBL2426 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Casein kinase I isoform delta CHEMBL2828 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Homeodomain-interacting protein kinase 4 CHEMBL1075167 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Serine/threonine-protein kinase MRCK alpha CHEMBL4516 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform CHEMBL2349 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 4 CHEMBL1075115 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma CHEMBL3829 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 5.2 | 5.2 | 6309.6 | 1 |
| Casein kinase I isoform gamma-3 CHEMBL5084 | Ki | 5.2 | 5.2 | 6309.6 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta CHEMBL2801 | Ki | 5.2 | 5.2 | 6309.6 | 1 |
| Casein kinase I isoform alpha CHEMBL2793 | Ki | 5.2 | 5.2 | 6309.6 | 1 |
| Mitogen-activated protein kinase 1 CHEMBL4040 | Ki | 5.1 | 5.1 | 7943.3 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 5.1 | 5.1 | 7943.3 | 1 |
| Protein kinase C zeta type CHEMBL3438 | Ki | 5.1 | 5.1 | 7943.3 | 1 |