Assay Detail
Functional
CHEMBL1964107
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: DYRK1A
1056
Total Activities
1037
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (CHEMBL2292) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1056 | 6.28 | 9.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1980407 | — | — | 1 | 9.40 |
| CHEMBL1965660 | — | — | 2 | 9.10 |
| CHEMBL1987448 | — | — | 1 | 9.10 |
| CHEMBL1992220 | — | — | 1 | 9.00 |
| CHEMBL1980995 | — | — | 1 | 8.60 |
| CHEMBL2001751 | — | — | 1 | 8.60 |
| CHEMBL2005509 | — | — | 1 | 8.60 |
| CHEMBL1996980 | — | — | 1 | 8.50 |
| CHEMBL1981133 | — | — | 1 | 8.50 |
| CHEMBL1966628 | — | — | 1 | 8.50 |
| CHEMBL1966524 | — | — | 1 | 8.40 |
| CHEMBL1967302 | — | — | 1 | 8.40 |
| CHEMBL1969588 | — | — | 1 | 8.40 |
| CHEMBL226403 | — | — | 1 | 8.40 |
| CHEMBL2000345 | — | — | 1 | 8.30 |
| CHEMBL2007574 | — | — | 1 | 8.30 |
| CHEMBL1976936 | — | — | 1 | 8.30 |
| CHEMBL1973098 | — | — | 1 | 8.20 |
| CHEMBL1983534 | — | — | 1 | 8.20 |
| CHEMBL1987261 | — | — | 1 | 8.20 |
| CHEMBL1994669 | — | — | 1 | 8.20 |
| CHEMBL1241473 | — | — | 1 | 8.20 |
| CHEMBL1999931 | — | — | 1 | 8.20 |
| CHEMBL1995813 | — | — | 1 | 8.10 |
| CHEMBL1987679 | — | — | 1 | 8.10 |
| CHEMBL1994241 | — | — | 1 | 8.10 |
| CHEMBL1973540 | — | — | 1 | 8.10 |
| CHEMBL1967887 | — | — | 1 | 8.00 |
| CHEMBL1982271 | — | — | 1 | 8.00 |
| CHEMBL2005718 | — | — | 1 | 8.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1980407 | — | Ki | = | 0.3981 | nM | 9.40 |
| CHEMBL1965660 | — | Ki | = | 0.7943 | nM | 9.10 |
| CHEMBL1987448 | — | Ki | = | 0.7943 | nM | 9.10 |
| CHEMBL1965660 | — | Ki | = | 0.7943 | nM | 9.10 |
| CHEMBL1992220 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL1980995 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL2001751 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL2005509 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL1981133 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1996980 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1966628 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL226403 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1966524 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1969588 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1967302 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL2000345 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL2007574 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1976936 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1994669 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1241473 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1973098 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1983534 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1987261 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1999931 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1994241 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1995813 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1973540 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1987679 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1982271 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1967887 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1984548 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL226471 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL2005718 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1986855 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1980253 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1966204 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL526133 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1972290 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1994438 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL2000354 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1977223 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL225519 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL2006933 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL2006439 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1996817 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1972339 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1682553 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1973720 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1980562 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1988581 | — | Ki | = | 25.12 | nM | 7.60 |